SCHEMBL8511475

SCHEMBL8511475

CC1(C)CCC(C)(C)c2cc(-c3cc(C4=CCNCC4)ccn3)ccc21

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
QDPR P09417 3/20 0.43
HTR2C P28335 8/20 0.40
SIGMAR1 Q99720 2/20 0.40
WNT3A P56704 1/20 0.39
LRRK2 Q5S007 1/20 0.38
ALK Q9UM73 1/20 0.37
RARA P10276 1/20 0.36
RARB P10826 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL8654933 0.90 WNT3A (0.40) QDPRHTR2CWNT3ARARARARB
SCHEMBL9612545 0.81 TGFBR1 (0.43) QDPRHTR2CSIGMAR1WNT3AALK
SCHEMBL18961191 0.80 RARA (0.47) RARARARB
SCHEMBL9612753 0.80 RARA (0.53) QDPRHTR2CSIGMAR1RARARARB
SCHEMBL8514545 0.76 HTR2C (0.38) QDPRHTR2CSIGMAR1ALKRARA
SCHEMBL8515364 0.75 QDPR (0.39) QDPRHTR2CSIGMAR1ALKRARA
Hydrochloric Acid SCHEMBL8534872 0.75 HTR2C (0.39) QDPRHTR2CSIGMAR1ALKRARA
SCHEMBL16998862 0.74 RARB (0.55) RARARARB
SCHEMBL8512658 0.74 RARA (0.44) RARARARB
SCHEMBL8515212 0.73 ALDH1A1 (0.42) QDPRRARARARB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO claimed
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed