SCHEMBL8511490

SCHEMBL8511490

CC1(C)CCC(C)(C)c2cc(-c3ccnc(N4CCN(C(=N)N)CC4)n3)ccc21

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DKK1 O94907 3/20 0.42
RARA P10276 1/20 0.41
RARB P10826 1/20 0.41
CA9 Q16790 5/20 0.40
CA2 P00918 3/20 0.40
PIK3CA P42336 2/20 0.40
PIK3CD O00329 1/20 0.40
PIK3R1 P27986 1/20 0.40
PIK3CB P42338 1/20 0.40
FAAH O00519 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
SCN9A Q15858 2/20 0.38
SORD Q00796 1/20 0.38
HCAR2 Q8TDS4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8515565 0.99 DKK1 (0.41) DKK1RARARARBCA9CA2
SCHEMBL9612771 0.90 RARA (0.41) DKK1RARARARBCA9CA2
Hydrochloric Acid SCHEMBL8667697 0.89 RARA (0.41) DKK1RARARARBCA9CA2
SCHEMBL8513704 0.85 RARA (0.40) DKK1RARARARBCA9CA2
SCHEMBL8513700 0.84 DKK1 (0.38) DKK1RARARARBCA9CA2
SCHEMBL8513698 0.84 DKK1 (0.38) DKK1RARARARBCA9CA2
SCHEMBL8510951 0.83 DKK1 (0.45) DKK1RARARARBPIK3CAPIK3CD
SCHEMBL8515365 0.82 RARA (0.33) DKK1RARARARBCA9CA2
Hydrochloric Acid SCHEMBL8512387 0.82 DKK1 (0.44) DKK1RARARARBPIK3CAPIK3CD
SCHEMBL8514868 0.81 DKK1 (0.64) DKK1RARARARBPIK3CAPIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO claimed
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed