SCHEMBL8513704

SCHEMBL8513704

CC1(C)CCC(C)(C)c2cc(-c3ccnc(N4CCN(C(=N)NC#N)CC4)n3)ccc21

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RARA P10276 1/20 0.40
RARB P10826 1/20 0.40
FAAH O00519 2/20 0.39
CA9 Q16790 5/20 0.38
CA2 P00918 3/20 0.38
PIK3CA P42336 1/20 0.37
DKK1 O94907 3/20 0.37
HCAR2 Q8TDS4 1/20 0.37
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
PANK3 Q9H999 1/20 0.36
DGAT1 O75907 1/20 0.35
CCNT1 O60563 1/20 0.35
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
CDK9 P50750 1/20 0.35
SORD Q00796 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9612771 0.86 RARA (0.41) RARARARBFAAHCA9CA2
Hydrochloric Acid SCHEMBL8667697 0.85 RARA (0.41) RARARARBFAAHCA9CA2
SCHEMBL8511490 0.85 DKK1 (0.42) RARARARBFAAHCA9CA2
Hydrochloric Acid SCHEMBL8515565 0.84 DKK1 (0.41) RARARARBFAAHCA9CA2
SCHEMBL8513698 0.82 DKK1 (0.38) RARARARBFAAHCA9CA2
SCHEMBL8513700 0.82 DKK1 (0.38) RARARARBFAAHCA9CA2
SCHEMBL8515120 0.77 DKK1 (0.38) RARARARBFAAHCA9CA2
SCHEMBL8515121 0.77 DKK1 (0.38) RARARARBFAAHCA9CA2
SCHEMBL8512407 0.77 ADRB1 (0.44) RARARARBPIK3CADKK1
SCHEMBL2015814 0.77 ACHE (0.52) RARARARBFAAHCA9CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO claimed
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed