SCHEMBL8515365

SCHEMBL8515365

C=C(C)c1ccc(-c2ccnc(N3CCN(C(=N)N)CC3)n2)cc1C(C)(C)C.CC1(C)CCC(C)(C)c2cc(-c3ccnc(-c4ccc(C(=N)N)cc4)n3)ccc21

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RARA P10276 1/20 0.33
RARB P10826 1/20 0.33
CA9 Q16790 3/20 0.31
CA2 P00918 2/20 0.31
TSHR P16473 1/20 0.31
DKK1 O94907 1/20 0.30
FAAH O00519 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8511972 0.87 DKK1 (0.39) CA9CA2TSHRDKK1FAAH
Hydrochloric Acid SCHEMBL8514429 0.86 DKK1 (0.38) CA9CA2TSHRDKK1FAAH
SCHEMBL8511490 0.82 DKK1 (0.42) RARARARBCA9CA2DKK1
Hydrochloric Acid SCHEMBL8515565 0.81 DKK1 (0.41) RARARARBCA9CA2DKK1
SCHEMBL8515254 0.77 RARB (0.51) RARARARB
SCHEMBL31060783 0.77 RARB (0.51) RARARARB
SCHEMBL9612771 0.76 RARA (0.41) RARARARBCA9CA2DKK1
Hydrochloric Acid SCHEMBL8667697 0.75 RARA (0.41) RARARARBCA9CA2DKK1
SCHEMBL8515183 0.73 ACHE (0.48) FAAH
SCHEMBL8512423 0.72 ADRB1 (0.42) DKK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO claimed