SCHEMBL8514935

SCHEMBL8514935

O=C(O)c1c(-c2ccc(Cc3ccc(OC(F)(F)F)cc3)cc2)[nH]c2ccccc2c1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.43
KIF11 P52732 1/20 0.42
FFAR1 O14842 1/20 0.41
FFAR4 Q5NUL3 1/20 0.41
HAT1 O14929 1/20 0.41
EP300 Q09472 1/20 0.41
SERPINE1 P05121 2/20 0.40
CDK8 P49336 1/20 0.40
NTRK3 Q16288 1/20 0.40
TDP1 Q9NUW8 2/20 0.39
KDM4E B2RXH2 1/20 0.39
STING1 Q86WV6 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
MAPK8 P45983 1/20 0.39
MAPK10 P53779 1/20 0.39
TRPV1 Q8NER1 1/20 0.39
SCN9A Q15858 1/20 0.38
CTSV O60911 1/20 0.38
CTSL P07711 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8613034 0.92 KIF11 (0.47) KIF11SERPINE1TDP1KDM4ESTING1
SCHEMBL8512623 0.87 NPC1 (0.47) KDM4EMAPTKMT2AMAPK10
SCHEMBL8514278 0.84 KIF11 (0.42) ESR1KIF11FFAR1FFAR4HAT1
SCHEMBL8532964 0.84 MAT2A (0.52) ESR1KIF11CDK8NTRK3TDP1
SCHEMBL8537609 0.84 KIF11 (0.44) ESR1KIF11CDK8NTRK3TDP1
SCHEMBL8512448 0.80 KMT2A (0.50) TDP1KDM4EMAPTKMT2AMAPK10
SCHEMBL7455829 0.77 TUBB4A (0.57) TDP1KDM4EMAPTKMT2A
SCHEMBL8537300 0.77 KIF11 (0.46) KIF11SERPINE1TDP1STING1MAPT
SCHEMBL6280799 0.76 KDM4E (0.59) ESR1TDP1KDM4EKMT2A
SCHEMBL8538008 0.76 CTSV (0.63) KIF11KDM4EKMT2ACTSVCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108697705-A combination product 利物浦热带医学院 2018-10-23 CN claimed
CN-108697705-A combination product 利物浦热带医学院 2018-10-23 CN disclosed
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed