SCHEMBL8537609

SCHEMBL8537609

O=c1c(Cl)c(-c2ccc(Cc3ccc(OC(F)(F)F)cc3)cc2)[nH]c2ccccc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.44
ESR1 P03372 1/20 0.39
MAT2A P31153 1/20 0.38
SLC6A4 P31645 1/20 0.38
CDK8 P49336 1/20 0.37
NTRK3 Q16288 1/20 0.37
HCRTR1 O43613 2/20 0.37
HCRTR2 O43614 2/20 0.37
CNR1 P21554 2/20 0.37
CTSV O60911 1/20 0.37
CTSL P07711 1/20 0.37
CHRM5 P08912 2/20 0.36
TACR1 P25103 1/20 0.36
PDE2A O00408 1/20 0.36
DHODH Q02127 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE10A Q9Y233 1/20 0.36
KDM4E B2RXH2 1/20 0.36
CRHBP P24387 1/20 0.36
CRHR2 Q13324 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8532964 0.86 MAT2A (0.52) KIF11ESR1MAT2ASLC6A4CDK8
SCHEMBL8514935 0.84 ESR1 (0.43) KIF11ESR1CDK8NTRK3CTSV
SCHEMBL8514278 0.84 KIF11 (0.42) KIF11ESR1MAT2ASLC6A4CDK8
SCHEMBL8535741 0.82 ABL1 (0.41) KIF11HCRTR1HCRTR2CHRM5
SCHEMBL8512623 0.81 NPC1 (0.47) HCRTR1KDM4EMAPTKMT2A
SCHEMBL8538008 0.78 CTSV (0.63) KIF11CTSVCTSLPDE10AKDM4E
SCHEMBL8537794 0.77 MAT2A (0.50) KIF11MAT2ASLC6A4CTSVCTSL
SCHEMBL8535303 0.77 MAT2A (0.55) KIF11MAT2ASLC6A4CNR1
SCHEMBL8515371 0.77 MAT2A (0.56) KIF11MAT2APDE2ADHODHPDE4B
SCHEMBL8537300 0.76 KIF11 (0.46) KIF11MAT2ATACR1PDE2ADHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO claimed
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed