SCHEMBL8515409

SCHEMBL8515409

CCOC(=O)Cc1ccc(B(O)OC(C)(C)C(C)(C)O)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.45
LMNA P02545 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
CYP4Z1 Q86W10 1/20 0.43
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TSHR P16473 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CYP4F2 P78329 1/20 0.37
CYP4A11 Q02928 1/20 0.37
TBXAS1 P24557 1/20 0.37
LIPE Q05469 1/20 0.37
FDFT1 P37268 1/20 0.37
GAA P10253 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
NPC1 O15118 1/20 0.35
PKM P14618 1/20 0.35
NFKB1 P19838 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28636456 0.84 MAPT (0.48) MAPTLMNASMN1; SMN2CYP4Z1KDM4E
SCHEMBL17315637 0.82 RXRA (0.42) LMNAKDM4EALDH1A1TSHRHSD17B10
SCHEMBL16278156 0.82 SMN1; SMN2 (0.36) MAPTLMNASMN1; SMN2KDM4EALDH1A1
SCHEMBL1997052 0.82 CA1 (0.49) MAPTLMNASMN1; SMN2ALDH1A1MEN1
SCHEMBL18705952 0.79 LPL (0.32)
SCHEMBL1239798 0.79 LPL (0.52) MAPTLMNASMN1; SMN2CYP4Z1KDM4E
SCHEMBL9986342 0.77 PPARG (0.37) TSHR
SCHEMBL68851 0.76 CYP4Z1 (0.62) MAPTLMNASMN1; SMN2CYP4Z1KDM4E
SCHEMBL1129027 0.76 LPL (0.32)
SCHEMBL1490590 0.76 F11 (0.47) SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2643291-A2 CALCIUM-SENSING RECEPTOR-ACTIVE COMPOUNDS Leo Pharma A/S (DK) 2013-10-02 EP disclosed
US-20130244995-A1 CALCIUM-SENSING RECEPTOR-ACTIVE COMPOUNDS LEO PHARMA A/S (DK) 2013-09-19 US disclosed
WO-2012069420-A2 CALCIUM-SENSING RECEPTOR-ACTIVE COMPOUNDS LEO PHARMA A/S (DK) 2012-05-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130244995-A1 CALCIUM-SENSING RECEPTOR-ACTIVE COMPOUNDS CASR, CALCR, PTH1R MAPT 3151/4885LMNA 2262/4885SMN1; SMN2 3811/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.