SCHEMBL8516504

SCHEMBL8516504

C=CCc1cccc(-c2ccnc(C#CC(C)O)n2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.41
CTSS P25774 4/20 0.34
CTSK P43235 3/20 0.34
KARS1 Q15046 2/20 0.32
KMO O15229 2/20 0.32
LMNA P02545 3/20 0.32
MAPT P10636 3/20 0.32
GAA P10253 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HTT P42858 1/20 0.32
DYRK1A Q13627 2/20 0.31
CLK4 Q9HAZ1 2/20 0.31
DYRK1B Q9Y463 1/20 0.31
MAPK1 P28482 1/20 0.31
MAP4K4 O95819 1/20 0.31
CTSL P07711 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8517692 0.83 ADRB2 (0.39) GAAMEN1KMT2AALDH1A1DYRK1A
SCHEMBL8517940 0.78 ASIC3 (0.36) PTGS2KMOLARS1
SCHEMBL19766402 0.73 KMO (0.39) PTGS2KARS1KMOLMNAMAPT
SCHEMBL8517808 0.72 ALDH1A1 (0.36) PTGS2LMNAMAPTGAASMN1; SMN2
SCHEMBL8517606 0.72 ASIC3 (0.35) KMOLMNADYRK1ACLK4DYRK1B
SCHEMBL3792469 0.72 PTGS2 (0.49) PTGS2CTSSCTSKKARS1LMNA
SCHEMBL7864423 0.68 CDK8 (0.43) PTGS2CTSKKMOMAPK1CTSL
SCHEMBL8517769 0.68 GABRA1 (0.39) PTGS2LMNAMAPTGAASMN1; SMN2
SCHEMBL9796794 0.67 HRH3 (0.52) PTGS2CTSSLMNASMN1; SMN2KDM4E
SCHEMBL29725141 0.67 HRH3 (0.52) PTGS2CTSSLMNASMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628530-B1 ACETYLENE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, LIQUID CRYSTAL COMPOSITION CONTAINING THE SAME AS ACTIVE INGREDIENT, AND LIQUID CRYSTAL ELEMENT MADE THEREFROM SUMITOMO CHEMICAL CO (JP) 1999-03-24 EP disclosed
US-5534188-A Acetylene derivatives, process for producing the same, liquid crystal composition containing the same as an active ingredient, and liquid crystal element using said liquid crystal composition SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1996-07-09 US disclosed
EP-0628530-A1 ACETYLENE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, LIQUID CRYSTAL COMPOSITION CONTAINING THE SAME AS ACTIVE INGREDIENT, AND LIQUID CRYSTAL ELEMENT MADE THEREFROM SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1994-12-14 EP disclosed