SCHEMBL8517870

SCHEMBL8517870

CC(C)(C)OC(=O)C(CCCN)(NCCC#N)C(=O)OC(C)(C)C

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
DGAT1 O75907 1/20 0.31
CTSS P25774 3/20 0.30
CTSK P43235 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7719979 0.78 TDP1 (0.48) MEN1KMT2A
SCHEMBL28165431 0.72 ITGB3 (0.34) DGAT1
SCHEMBL29454707 0.68 DGAT1 (0.34) MEN1KMT2ADGAT1
SCHEMBL8611222 0.68 MEN1 (0.39) MEN1KMT2ADGAT1CTSSCTSK
SCHEMBL16411264 0.67 DGAT1 (0.33) DGAT1
SCHEMBL8797158 0.67 DGAT1 (0.38) DGAT1
SCHEMBL3294151 0.67 DGAT1 (0.38) DGAT1
SCHEMBL27831974 0.66 MEN1 (0.37) MEN1KMT2ADGAT1CTSSCTSK
SCHEMBL13305942 0.65 MEN1 (0.38) MEN1KMT2ADGAT1
SCHEMBL1304101 0.65 TDP1 (0.53) MEN1KMT2ACTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6001824-A Butyryl-tyrosinyl spermine, analogs thereof and methods of preparing and using same THE TRUSTEES OF COLUMBIA UNIVERSITY (US) 1999-12-14 US disclosed
WO-1996022962-A1 BUTYRYL-TYROSINYL SPERMINE, ANALOGS THEREOF AND METHODS OF PREPARING AND USING SAME THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 1996-08-01 WO disclosed