SCHEMBL8520072

SCHEMBL8520072

C1=COc2c(cccc2N2CCN(CCCC3(Cc4ccccc4)CCC3)CC2)O1

nearest known ligand 0.48

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.48
DRD2 P14416 2/20 0.41
HTR7 P34969 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9466376 0.77 HTR1A (0.56) HTR1ADRD2
SCHEMBL9175441 0.72 HTR1A (0.57) HTR1ADRD2
SCHEMBL7812155 0.68 DRD2 (0.49) HTR1ADRD2
SCHEMBL8303446 0.66 HTR1A (0.93) HTR1ADRD2
SCHEMBL9176466 0.65 SLC6A2 (0.37) HTR1AHTR7
SCHEMBL7534943 0.63 ADRB1 (0.62) HTR1ADRD2HTR7
SCHEMBL9181453 0.62 KMT2A (0.41)
SCHEMBL9722314 0.62 MAOA (0.40)
SCHEMBL156160 0.61 MAOA (0.54)
SCHEMBL7134969 0.61 TSHR (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5990114-A ADMINISTERING 1,4-SUBSTITUTED PIPERAZINE DERIVATIVES OF GIVEN FORMULA TO TREAT NEUROMUSCULAR DYSFUNCTION OF THE LOWER URINARY TRACT; BOTH PRE- AND POST-SYNAPTIC ANTAGONISM; SUCH AS 1-(2-((2-PYRIDYLAMINO)ETHYL)-4-(4-INDOLYL)PIPERAZINE RECORDATI, S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1999-11-23 US disclosed