SCHEMBL8520543

SCHEMBL8520543

C=CCn1c(C)c2c(c1C)C(=O)C(C)=C(C)C2=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.48
NPSR1 Q6W5P4 1/20 0.39
KMT2A Q03164 4/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
MEN1 O00255 2/20 0.38
KDM4E B2RXH2 2/20 0.38
HPGD P15428 2/20 0.38
GAA P10253 1/20 0.34
CNR2 P34972 1/20 0.34
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
MAPT P10636 1/20 0.33
ALDH1A1 P00352 3/20 0.33
KDM4C Q9H3R0 1/20 0.33
NPC1 O15118 1/20 0.33
TP53 P04637 1/20 0.33
CYP2C19 P33261 1/20 0.33
RAB9A P51151 1/20 0.33
ADORA2B P29275 1/20 0.33
USP2 O75604 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8437874 0.73 KDM4E (0.39) CYP3A4KMT2ASMN1; SMN2MEN1KDM4E
SCHEMBL8437857 0.70 PTGS2 (0.39) CYP3A4SMN1; SMN2KDM4EHPGDCYP1A2
SCHEMBL8434025 0.68 PTGS2 (0.48) KMT2AMEN1KDM4EGAAMAPT
SCHEMBL28662 0.66 CYP3A4 (1.00) CYP3A4NPSR1KMT2ASMN1; SMN2MEN1
SCHEMBL4622249 0.65 CYP3A4 (0.46) CYP3A4NPSR1KMT2ASMN1; SMN2MEN1
SCHEMBL8640814 0.65 KMT2A (0.43) CYP3A4NPSR1KMT2ASMN1; SMN2MEN1
SCHEMBL5391867 0.64 CYP3A4 (0.45) CYP3A4NPSR1KMT2ASMN1; SMN2MEN1
SCHEMBL9818017 0.64 CASP3 (0.47) CYP3A4KMT2ASMN1; SMN2MEN1KDM4E
SCHEMBL10997976 0.62 CYP3A4 (0.79) CYP3A4NPSR1KMT2ASMN1; SMN2MEN1
SCHEMBL9246057 0.62 CYP3A4 (0.76) CYP3A4NPSR1KMT2ASMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5889185-A Method of synthesizing isoindolequinones and derivatives thereof THE UNIVERSITY OF AKRON (US) 1999-03-30 US disclosed
WO-1998046567-A1 METHOD OF SYNTHESIZING ISOINDOLEQUINONES AND DERIVATIVES THEREOF THE UNIVERSITY OF AKRON (US) 1998-10-22 WO disclosed