SCHEMBL8523477

SCHEMBL8523477

CC(C)c1ccc(-n2nc3c([nH]c(=O)c4ccccc43)c2O)cc1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PBK Q96KB5 8/20 0.39
DHODH Q02127 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
ADRA1B P35368 1/20 0.36
PARP1 P09874 3/20 0.35
DHFR P00374 1/20 0.35
ADORA3 P0DMS8 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8522571 0.81 ADORA3 (0.47) RAB9AMAPTPARP1ADORA3
SCHEMBL8523766 0.77 KDM4E (0.39) DHODHSMN1; SMN2NPC1RAB9AMAPT
SCHEMBL4057758 0.70 RAB9A (0.51) DHODHSMN1; SMN2NPC1RAB9AALDH1A1
Water SCHEMBL8326247 0.69 ESR2 (0.33) DHODHSMN1; SMN2ALDH1A1LMNA
SCHEMBL4059604 0.64 RAB9A (0.55) DHODHSMN1; SMN2NPC1RAB9AALDH1A1
SCHEMBL8324852 0.63 GAA (0.53) SMN1; SMN2NPC1RAB9ALMNAADORA3
SCHEMBL5324211 0.62 SMN1; SMN2 (0.71) SMN1; SMN2NPC1RAB9ATP53ALDH1A1
SCHEMBL23400622 0.61 LMNA (0.54) SMN1; SMN2NPC1RAB9ATP53MAPT
SCHEMBL22093797 0.60 MAT2A (0.80) MAPTALDH1A1LMNADHFR
SCHEMBL31145413 0.60 MAT2A (0.80) MAPTALDH1A1LMNADHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888347-A1 PHARMACEUTICALLY USEFUL COMPOUNDS Astra Pharmaceuticals Limited (GB) 1999-01-07 EP claimed
WO-1997034893-A1 PHARMACEUTICALLY USEFUL COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-09-25 WO claimed