SCHEMBL8527896

SCHEMBL8527896

CC(C)(C)[Si](C)(C)OCC(CC=Cc1cccnc1)CC(C(=O)O)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.42
CHRNA4 P43681 2/20 0.42
TBXAS1 P24557 2/20 0.38
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34
JUN P05412 1/20 0.34
MAPT P10636 1/20 0.34
NFKB1 P19838 1/20 0.34
MAPK1 P28482 1/20 0.34
RAB9A P51151 1/20 0.34
GPR55 Q9Y2T6 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNA7 P36544 1/20 0.34
MEN1 O00255 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
ALOX15 P16050 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8527898 0.80 TBXAS1 (0.39) CHRNB2CHRNA4TBXAS1CYP11B1CYP11B2
SCHEMBL8528974 0.74 TBXAS1 (0.46) CHRNB2CHRNA4TBXAS1KDM4ENPC1
SCHEMBL9843049 0.74 TBXAS1 (0.47) CHRNB2CHRNA4TBXAS1KDM4ENPC1
SCHEMBL9843054 0.74 TBXAS1 (0.47) CHRNB2CHRNA4TBXAS1KDM4ENPC1
SCHEMBL16798382 0.73 CYP2C19 (0.42) MAPK1MEN1CYP2D6CYP2C19KMT2A
SCHEMBL8668533 0.70 CHRNB2 (0.41) CHRNB2CHRNA4TBXAS1CYP11B1CYP11B2
SCHEMBL9733096 0.70 TBXAS1 (0.41) CHRNB2CHRNA4TBXAS1KDM4ENPC1
SCHEMBL9733100 0.70 TBXAS1 (0.41) CHRNB2CHRNA4TBXAS1KDM4ENPC1
SCHEMBL10618822 0.69 TBXAS1 (0.48) CHRNB2CHRNA4TBXAS1CYP11B1CYP11B2
SCHEMBL10618801 0.69 TBXAS1 (0.48) CHRNB2CHRNA4TBXAS1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5849922-A Preparation of substituted alkenoic acids ELI LILLY AND COMPANY (US) 1998-12-15 US disclosed
US-5849766-A Carbamoyl substituted heterocycles ELI LILLY AND COMPANY (US) 1998-12-15 US disclosed