SCHEMBL8531874

SCHEMBL8531874

Cc1cc2c(cc1C)C(=O)C(CC(=O)N1C(C)CCC1C)CC2

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.36
CYP26A1 O43174 5/20 0.36
CYP24A1 Q07973 2/20 0.36
ITGB3 P05106 3/20 0.35
ITGA2B P08514 3/20 0.35
TSHR P16473 1/20 0.34
CHRM2 P08172 2/20 0.34
CHRM4 P08173 2/20 0.34
CHRM1 P11229 2/20 0.34
CHRM3 P20309 2/20 0.34
CYP19A1 P11511 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GLA P06280 1/20 0.33
HPGD P15428 1/20 0.33
ACHE P22303 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8534988 0.83 CYP11B1 (0.41) DGAT1CYP26A1TSHRCHRM2CHRM4
SCHEMBL8534684 0.82 DGAT1 (0.50) DGAT1CYP26A1CYP24A1ITGB3ITGA2B
SCHEMBL8533781 0.75 ROCK2 (0.38) CYP26A1CYP24A1
SCHEMBL11723357 0.72 THRA (0.52)
SCHEMBL8535491 0.71 IMPDH2 (0.40) CYP26A1CYP24A1CYP19A1
Hydrochloric Acid SCHEMBL8531523 0.71 METAP1 (0.54)
Iodide SCHEMBL8534944 0.71 CYP26A1 (0.39) CYP26A1CYP24A1CYP19A1
SCHEMBL8531913 0.68 CHRM2 (0.48) DGAT1CYP26A1TSHRCHRM2CHRM4
SCHEMBL8532323 0.68 CHRM2 (0.46) TSHRCHRM2CHRM4CHRM1CHRM3
SCHEMBL8536553 0.66 DGAT1 (0.57) DGAT1CYP26A1CYP24A1ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5847159-A 1- ω-(3,4-dihydro-2-naphthalenyl)alkyl!-cyclic amine derivatives, process for preparing the same, and pharmaceutical composition containing the same DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1998-12-08 US disclosed
EP-0825180-A1 1-OMEGA-(3,4-DIHYDRO-2-NAPHTHALENYL)ALKYL] CYCLIC AMINE DERIVATIVES, PROCESS FOR PRODUCING THE SAME, AND MEDICINAL COMPOSITION CONTAINING THE SAME DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1998-02-25 EP disclosed