SCHEMBL8534140

SCHEMBL8534140

COc1ccc2c(=O)cc(-c3cnn(Cc4ccc(OC(F)(F)F)cc4)c3)[nH]c2c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
MAT2A P31153 1/20 0.42
HPGD P15428 7/20 0.41
KDM4E B2RXH2 6/20 0.41
SMN1; SMN2 Q16637 4/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
ADORA2A P29274 1/20 0.41
ADORA2B P29275 1/20 0.41
ADORA1 P30542 1/20 0.41
LMNA P02545 3/20 0.40
CHRM5 P08912 3/20 0.40
MAPT P10636 1/20 0.40
MAPK1 P28482 1/20 0.39
KLKB1 P03952 1/20 0.38
CYP19A1 P11511 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8534905 0.88 CTSV (0.47) ALDH1A1KMT2AHPGDKDM4ESMN1; SMN2
SCHEMBL8538579 0.84 MAT2A (0.61) MAT2AADORA2AADORA2BADORA1CHRM5
SCHEMBL8533234 0.75 MAT2A (0.49) MAT2AADORA2AADORA2BADORA1CHRM5
SCHEMBL8653277 0.75 MAT2A (0.49) MAT2AADORA2AADORA2BADORA1CHRM5
SCHEMBL9607232 0.74 ABL1 (0.42) ALDH1A1HPGDKDM4ESMN1; SMN2ADORA2A
SCHEMBL8536122 0.73 CTSV (0.60) ALDH1A1KMT2AHPGDKDM4ERAB9A
SCHEMBL8513871 0.72 MAT2A (0.46) MAT2AADORA2AADORA2BADORA1CHRM5
SCHEMBL18097397 0.72 PDE2A (0.47) CHRM5KLKB1
SCHEMBL8537370 0.72 MAT2A (0.43) MEN1KMT2AMAT2AADORA2AADORA2B
SCHEMBL8536502 0.72 MAT2A (0.43) ALDH1A1MEN1KMT2AMAT2AADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO claimed
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed
WO-2012069856-A1 ANTIMALARIAL COMPOUNDS LIVERPOOL SCHOOL OF TROPICAL MEDICINE (GB) 2012-05-31 WO disclosed