SCHEMBL8540730

SCHEMBL8540730

CSCc1cc(Br)ccc1-c1ncc[nH]1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MC4R P32245 2/20 0.46
ADRA2A P08913 2/20 0.43
ADRA2B P18089 2/20 0.43
ADRA2C P18825 2/20 0.43
NISCH Q9Y2I1 2/20 0.36
ALDH1A1 P00352 2/20 0.35
MTOR P42345 1/20 0.34
ADK P55263 1/20 0.34
FPR2 P25090 5/20 0.34
CSNK1A1 P48729 1/20 0.33
TYRO3 Q06418 1/20 0.33
DYRK1B Q9Y463 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP19A1 P11511 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8537559 0.91 MC4R (0.44) MC4RADRA2AADRA2BADRA2CNISCH
SCHEMBL8540790 0.84 NISCH (0.37) MC4RADRA2ANISCHALDH1A1MTOR
SCHEMBL8540597 0.82 CSNK1A1 (0.36) MC4RNISCHALDH1A1MTORADK
SCHEMBL8541400 0.82 MC4R (0.37) MC4RNISCHALDH1A1MTORADK
SCHEMBL8536816 0.82 JAK2 (0.47) MC4RNISCHALDH1A1MTORADK
SCHEMBL8537087 0.80 CSNK1A1 (0.45) MC4RADRA2AADRA2BADRA2CNISCH
SCHEMBL8539649 0.80 NOS3 (0.47) MC4RADRA2AADRA2CNISCHALDH1A1
SCHEMBL8541205 0.79 NISCH (0.36) MC4RADRA2AADRA2BADRA2CNISCH
SCHEMBL8535625 0.79 NISCH (0.49) ADRA2ANISCHALDH1A1MTORADK
SCHEMBL8539601 0.79 CYP19A1 (0.41) NISCHMTORADKCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0857171-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1998-08-12 EP disclosed
WO-1997015555-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1997-05-01 WO disclosed