SCHEMBL8537871

SCHEMBL8537871

CC(=O)OCCn1cnc2c(Cl)nc(Nc3ccccc3)nc21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.42
HDAC2 Q92769 3/20 0.42
HDAC8 Q9BY41 2/20 0.42
HDAC6 Q9UBN7 2/20 0.42
YTHDC1 Q96MU7 1/20 0.41
TK1 P04183 1/20 0.41
CDK4 P11802 1/20 0.40
CCND1 P24385 1/20 0.40
CCND2 P30279 1/20 0.40
CCND3 P30281 1/20 0.40
ABL1 P00519 1/20 0.40
BTK Q06187 1/20 0.40
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.39
MAPK1 P28482 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
ADORA2B P29275 1/20 0.39
TMIGD3 P0DMS9 1/20 0.39
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8539832 0.93 TK1 (0.46) HDAC1HDAC2HDAC8HDAC6YTHDC1
SCHEMBL6523725 0.87 KDM4E (0.48) HDAC1HDAC2HDAC8HDAC6YTHDC1
SCHEMBL8539778 0.86 CDK1 (0.49) LMNAMAPK1
SCHEMBL8538543 0.81 HDAC1 (0.52) HDAC1HDAC2HDAC8HDAC6YTHDC1
SCHEMBL12537333 0.80 P2RX7 (0.50) HDAC1HDAC2HDAC8HDAC6YTHDC1
SCHEMBL8537887 0.78 TK1 (0.68) TK1
SCHEMBL5801330 0.78 HDAC3 (0.40) HDAC1HDAC2HDAC8HDAC6
SCHEMBL19553815 0.73 CNR2 (0.42) HDAC1HDAC2HDAC8HDAC6TK1
SCHEMBL19690966 0.73 CDK1 (0.45)
SCHEMBL8157896 0.73 CTSL (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0794781-A4 DRUGS TO PREVENT RECURRENT HERPES VIRUS INFECTIONS UNIV MASSACHUSETTS MEDICAL (US) 1998-04-22 EP disclosed
EP-0794781-A1 DRUGS TO PREVENT RECURRENT HERPES VIRUS INFECTIONS UNIVERSITY OF MASSACHUSETTS MEDICAL CENTER (US) 1997-09-17 EP disclosed
US-5646155-A ADMINISTERING A 9-SUBSTITUTED-N2-PHENYLGUANINE DERIVATIVE UNIVERSITY OF MASSACHUSETTS MEDICAL CENTER (US) 1997-07-08 US disclosed
WO-1996020711-A1 DRUGS TO PREVENT RECURRENT HERPES VIRUS INFECTIONS UNIVERSITY OF MASSACHUSETTS MEDICAL CENTER (US) 1996-07-11 WO disclosed