(3R)-Dunnione

(3R)-Dunnione

SCHEMBL8538701

CC1OC2=C(C(=O)C(=O)c3ccccc32)C1(C)C.CC1OC2=C(C(=O)C(=O)c3ccccc32)C1(C)C.c1ccc2[nH]c(-c3cscn3)nc2c1.c1ccc2[nH]c(-c3cscn3)nc2c1

nearest known ligand 0.55

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
METAP1 P53582 8/20 0.55
METAP2 P50579 5/20 0.55
NPC1 O15118 3/20 0.55
RAB9A P51151 2/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
KDM4E B2RXH2 1/20 0.55
TP53 P04637 1/20 0.55
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
ADORA3 P0DMS8 1/20 0.55
CYP2D6 P10635 1/20 0.55
TSHR P16473 1/20 0.55
CYP2C19 P33261 1/20 0.55
FKBP1A P62942 1/20 0.55
HIF1A Q16665 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
HDAC6 Q9UBN7 1/20 0.55
IDO1 P14902 2/20 0.47
TDO2 P48775 1/20 0.47
NQO1 P15559 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
(3R)-Dunnione SCHEMBL8535310 0.75 NQO1 (0.47) RAB9ASMN1; SMN2KDM4ETP53CYP1A2
Thiabendazole SCHEMBL29370729 0.74 METAP1 (1.00) METAP1METAP2NPC1RAB9ASMN1; SMN2
(3R)-Dunnione SCHEMBL29468606 0.74 NQO1 (0.63) NPC1RAB9ASMN1; SMN2KDM4ETP53
Thiabendazole SCHEMBL19842 0.74 METAP1 (1.00) METAP1METAP2NPC1RAB9ASMN1; SMN2
Thiabendazole SCHEMBL625588 0.74 METAP1 (1.00) METAP1METAP2NPC1RAB9ASMN1; SMN2
(3R)-Dunnione SCHEMBL103115 0.74 NQO1 (0.63) NPC1RAB9ASMN1; SMN2KDM4ETP53
(3R)-Dunnione SCHEMBL8535192 0.73 NQO1 (0.44) NPC1RAB9ASMN1; SMN2KDM4ECYP1A2
Thiabendazole SCHEMBL9856779 0.73 METAP1 (0.97) METAP1METAP2NPC1RAB9ASMN1; SMN2
Thiabendazole SCHEMBL11218788 0.73 METAP1 (0.97) METAP1METAP2NPC1RAB9ASMN1; SMN2
Thiabendazole SCHEMBL7733801 0.73 METAP1 (0.97) METAP1METAP2NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0861028-A1 FUNGICIDAL COMPOUNDS (B) BTG INTERNATIONAL LIMITED (GB) 1998-09-02 EP disclosed
WO-1997016970-A1 FUNGICIDAL COMPOUNDS (B) BRITISH TECHNOLOGY GROUP LIMITED (GB) 1997-05-15 WO disclosed