SCHEMBL8539360

SCHEMBL8539360

O=Cc1cc([N+](=O)[O-])ccc1-c1ncc[nH]1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.49
CYP3A4 P08684 2/20 0.44
NAMPT P43490 1/20 0.44
XDH P47989 1/20 0.44
NPC1 O15118 4/20 0.43
RAB9A P51151 3/20 0.43
MEN1 O00255 1/20 0.43
HSP90AA1 P07900 1/20 0.43
AGTR1 P30556 1/20 0.43
KMT2A Q03164 1/20 0.43
PTPN1 P18031 1/20 0.41
MAPT P10636 3/20 0.40
PARP1 P09874 1/20 0.40
KDM4E B2RXH2 1/20 0.40
METAP1 P53582 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ALDH1A1 P00352 2/20 0.40
PKN1 Q16512 1/20 0.40
PKN2 Q16513 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8539529 0.81 GPR35 (0.49) ERN1CYP3A4NAMPTXDHNPC1
SCHEMBL5249670 0.81 MAPT (0.56) CYP3A4NAMPTXDHNPC1RAB9A
SCHEMBL8536767 0.81 CYP3A4 (0.46) CYP3A4NAMPTXDHNPC1RAB9A
SCHEMBL5747525 0.79 MEN1 (0.46) CYP3A4NAMPTXDHNPC1RAB9A
SCHEMBL31463535 0.79 AMY1A (0.48) CYP3A4NAMPTXDHNPC1RAB9A
SCHEMBL8540776 0.79 AMY1A (0.48) CYP3A4NAMPTXDHNPC1RAB9A
SCHEMBL31098731 0.79 ERN1 (0.67) ERN1CYP3A4MEN1KMT2APTPN1
SCHEMBL12798324 0.79 ERN1 (0.67) ERN1CYP3A4MEN1KMT2APTPN1
SCHEMBL4055359 0.78 HSD17B10 (0.49) CYP3A4NAMPTXDHNPC1RAB9A
SCHEMBL9292469 0.78 NPC1 (0.44) CYP3A4NAMPTXDHNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0857171-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1998-08-12 EP disclosed
WO-1997015555-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1997-05-01 WO disclosed