SCHEMBL8540237

SCHEMBL8540237

C=CCN(CCc1ccccc1OCc1ccccc1)C(=O)OC(C)(C)C

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BCHE P06276 11/20 0.52
PTGER1 P34995 2/20 0.46
PTGER4 P35408 2/20 0.46
PTGER3 P43115 2/20 0.46
PTGER2 P43116 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.45
HTR1A P08908 1/20 0.45
DRD2 P14416 1/20 0.45
ABCB1 P08183 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8542129 0.90 PTGER1 (0.47) BCHEPTGER1PTGER4PTGER3PTGER2
SCHEMBL4521331 0.85 L3MBTL1 (0.47) BCHEL3MBTL1
SCHEMBL7825818 0.85 LTB4R (0.51) BCHEL3MBTL1
SCHEMBL7646792 0.82 HTR1A (0.51) BCHEPTGER1PTGER4PTGER3PTGER2
SCHEMBL4512033 0.79 TAAR1 (0.43) L3MBTL1
SCHEMBL19153323 0.77 HDAC3 (0.52) L3MBTL1
SCHEMBL1845821 0.75 HTR1A (0.48) PTGER1PTGER4PTGER3PTGER2L3MBTL1
SCHEMBL4520986 0.75 REN (0.37) L3MBTL1DRD2
SCHEMBL7835952 0.75 LTB4R (0.52) BCHEL3MBTL1
SCHEMBL4519565 0.74 TAAR1 (0.45) L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0815105-A1 HETEROCYCLIC SUBSTITUTED PIPERAZINONE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS HOECHST MARION ROUSSEL, INC. (US) 1998-01-07 EP disclosed
WO-1996028441-A1 HETEROCYCLIC SUBSTITUTED PIPERAZINONE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS HOECHST MARION ROUSSEL, INC. (US) 1996-09-19 WO disclosed