SCHEMBL8540815

SCHEMBL8540815

COCCNC(=O)Oc1ccc2[nH]cc(CCCCCl)c2c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 3/20 0.59
TRPV1 Q8NER1 3/20 0.56
MTNR1A P48039 6/20 0.54
MTNR1B P49286 5/20 0.54
LTA4H P09960 1/20 0.53
PLA2G2A P14555 1/20 0.53
KDM4E B2RXH2 2/20 0.52
HTR1A P08908 2/20 0.52
KMT2A Q03164 2/20 0.52
HSD17B10 Q99714 2/20 0.52
MEN1 O00255 1/20 0.52
ALDH1A1 P00352 1/20 0.52
CYP1A1 P04798 1/20 0.52
MPO P05164 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
HPGD P15428 1/20 0.52
NQO2 P16083 1/20 0.52
HTR2B P41595 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8537746 0.85 FAAH (0.54) FAAHTRPV1MTNR1AMTNR1BHTR1A
SCHEMBL9261940 0.84 KMT2A (0.57) TRPV1KMT2AHSD17B10MEN1RAB9A
SCHEMBL8557152 0.84 MTNR1A (0.56) MTNR1AMTNR1BKDM4EHTR1AKMT2A
SCHEMBL8539238 0.82 FAAH (0.51) FAAHTRPV1MTNR1AMTNR1BHTR1A
SCHEMBL9828299 0.82 HTR1D (0.67) MTNR1AMTNR1BKDM4EHTR1AKMT2A
SCHEMBL8540082 0.82 HTR2A (0.53) FAAHTRPV1MTNR1AMTNR1BHTR1A
SCHEMBL9698973 0.82 FAAH (0.57) FAAHTRPV1MTNR1AMTNR1BLTA4H
SCHEMBL8557536 0.80 MTNR1A (0.57) MTNR1AMTNR1BKDM4EHTR1AKMT2A
SCHEMBL9697617 0.80 HTR1D (0.57) MTNR1AMTNR1BKDM4EHTR1AKMT2A
SCHEMBL8544427 0.80 ADRA2A (0.71)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0496222-B1 Indole derivatives MERCK PATENT GMBH (DE) 1998-09-09 EP disclosed
EP-0496222-A1 Indole derivatives MERCK PATENT GmbH (DE) 1992-07-29 EP disclosed