SCHEMBL8543259

SCHEMBL8543259

Cc1nc(Cl)c(Cl)n1CCC1CCN(C(=O)CCc2ccccc2)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.50
GRIN2B Q13224 1/20 0.49
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48
FAAH O00519 1/20 0.48
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
NPC1 O15118 2/20 0.46
TDP1 Q9NUW8 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
USP19 O94966 1/20 0.44
CPB1 P15086 1/20 0.44
HPGD P15428 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
MAPT P10636 1/20 0.44
CHRNB2 P17787 1/20 0.44
CHRNB4 P30926 1/20 0.44
CHRNA3 P32297 1/20 0.44
CHRNA4 P43681 1/20 0.44
FKBP1A P62942 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8538799 0.84 PDE4B (0.53) POLBGRIN2BKDM4EALDH1A1FAAH
SCHEMBL8539033 0.83 HDAC3 (0.48) ALDH1A1FAAHMEN1KMT2A
SCHEMBL8696372 0.81 NPC1 (0.52) ALDH1A1MEN1KMT2ANPC1TDP1
SCHEMBL8542109 0.81 HRH3 (0.51) GRIN2BMEN1KMT2ATSHR
SCHEMBL8546968 0.77 F10 (0.57) POLBGRIN2BKDM4EALDH1A1FAAH
SCHEMBL8539110 0.77 FAAH (0.64) POLBGRIN2BKDM4EALDH1A1FAAH
SCHEMBL8541862 0.76 POLB (0.66) POLBGRIN2BKDM4EALDH1A1FAAH
SCHEMBL8544779 0.76 GRIN2B (0.60) POLBGRIN2BKDM4EALDH1A1FAAH
SCHEMBL8545014 0.75 CPB1 (0.60) POLBGRIN2BKDM4EALDH1A1FAAH
SCHEMBL8544549 0.75 GRIN2B (0.53) POLBGRIN2BKDM4EALDH1A1FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705258-B1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY KNOLL AG (DE) 1998-12-30 EP disclosed
EP-0705258-A1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY Knoll AG (DE) 1996-04-10 EP disclosed
WO-1995000507-A1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY KNOLL AG (DE) 1995-01-05 WO disclosed