SCHEMBL8538799

SCHEMBL8538799

Cc1nc2ccccc2n1CCC1CCN(C(=O)CCc2ccccc2)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 1/20 0.53
POLB P06746 2/20 0.50
GRIN2B Q13224 1/20 0.49
KDM4E B2RXH2 2/20 0.48
ALDH1A1 P00352 1/20 0.48
FAAH O00519 1/20 0.48
PDE6D O43924 1/20 0.48
BCHE P06276 2/20 0.47
ACHE P22303 2/20 0.47
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
NPC1 O15118 2/20 0.46
TDP1 Q9NUW8 1/20 0.46
BRD4 O60885 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
TNF P01375 1/20 0.45
LMNA P02545 2/20 0.45
TSHR P16473 1/20 0.45
HTT P42858 1/20 0.45
HRH3 Q9Y5N1 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9036480 0.87 P2RX3 (0.43) PDE4BPOLBGRIN2BKDM4EALDH1A1
SCHEMBL8543259 0.84 POLB (0.50) POLBGRIN2BKDM4EALDH1A1FAAH
SCHEMBL8541861 0.81 P2RX7 (0.53) GRIN2BTNFLMNAHRH3
SCHEMBL8136777 0.79 GRIN2B (0.49) PDE4BPOLBGRIN2BKDM4EALDH1A1
SCHEMBL8542324 0.79 HTT (0.58) PDE4BPOLBGRIN2BKDM4EALDH1A1
SCHEMBL8546968 0.77 F10 (0.57) POLBGRIN2BKDM4EALDH1A1FAAH
SCHEMBL2468538 0.77 USP19 (0.52) PDE4BMEN1KMT2ANPC1TDP1
SCHEMBL8544779 0.76 GRIN2B (0.60) POLBGRIN2BKDM4EALDH1A1FAAH
SCHEMBL8544549 0.75 GRIN2B (0.53) POLBGRIN2BKDM4EALDH1A1FAAH
SCHEMBL8545014 0.75 CPB1 (0.60) POLBGRIN2BKDM4EALDH1A1FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705258-B1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY KNOLL AG (DE) 1998-12-30 EP disclosed
US-5741800-A ANTIINFLAMMATORY AGENT, ANTIALLERGENS KNOLL AKTIENGESELLACHAFT (DE) 1998-04-21 US disclosed
EP-0705258-A1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY Knoll AG (DE) 1996-04-10 EP disclosed
WO-1995000507-A1 AZOLYL-CYCLIC AMINE DERIVATIVES WITH IMMUNOMODULATORY ACTIVITY KNOLL AG (DE) 1995-01-05 WO disclosed