SCHEMBL8544796

SCHEMBL8544796

O=C1CCc2cc(C(O)CCN3CCCCC3Cc3ccc(F)cc3)c(Cl)cc2N1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A2 O94788 2/20 0.35
ATM Q13315 4/20 0.35
CACNA1G O43497 2/20 0.35
METAP2 P50579 4/20 0.34
KCNH2 Q12809 3/20 0.34
DRD2 P14416 1/20 0.34
DRD3 P35462 1/20 0.34
GRIN1 Q05586 1/20 0.33
GRIN2B Q13224 1/20 0.33
CCR3 P51677 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27458015 0.85 ATM (0.33) ATMCACNA1GGRIN2BCCR3
SCHEMBL8544706 0.83 GRIN2B (0.40) GRIN2B
SCHEMBL8543058 0.82 CACNA1G (0.37) ALDH1A2ATMCACNA1GMETAP2DRD2
SCHEMBL8547312 0.75 MAOA (0.54) DRD2DRD3GRIN1GRIN2B
SCHEMBL8544708 0.72 GRIN2B (0.45) GRIN2BCCR3
SCHEMBL8545326 0.72 GRIN2B (0.45) GRIN2BCCR3
SCHEMBL8545330 0.72 GRIN2B (0.45) GRIN2BCCR3
SCHEMBL8541676 0.69 GRIN2B (0.56) ATMKCNH2GRIN2B
SCHEMBL8540835 0.69 GRIN2B (0.51) DRD2GRIN1GRIN2B
SCHEMBL27486618 0.68 ALDH1A1 (0.36) CACNA1GCCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0709384-B1 Benzylpiperidine derivatives having high affinity for binding sites of aminoacid receptors MERCK PATENT GMBH (DE) 1998-12-23 EP disclosed
US-5698553-A Benzylpiperidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-12-16 US disclosed
EP-0709384-A1 Benzylpiperidine derivatives having high affinity for binding sites of aminoacid receptors MERCK PATENT GmbH (DE) 1996-05-01 EP disclosed