SCHEMBL8548581

SCHEMBL8548581

CC(=O)NC1CCCc2c(ccc(OCc3ccccc3)c2OCc2ccccc2)C1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
ACHE P22303 1/20 0.47
MTNR1A P48039 3/20 0.47
MTNR1B P49286 3/20 0.47
MEN1 O00255 1/20 0.47
ALDH1A1 P00352 1/20 0.47
KMT2A Q03164 1/20 0.47
SGMS2 Q8NHU3 1/20 0.46
AGTR2 P50052 3/20 0.43
ACACB O00763 1/20 0.43
BRD4 O60885 3/20 0.43
TAOK1 Q7L7X3 2/20 0.41
TAOK3 Q9H2K8 2/20 0.41
PTPN1 P18031 1/20 0.41
AGTR1 P30556 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8547546 0.88 CA1 (0.46) CA1CA2ACHEMTNR1AMTNR1B
SCHEMBL8549143 0.78 ADRA1A (0.42) AGTR2AGTR1
SCHEMBL22681381 0.76 DRD2 (0.59) CA1CA2ACHEMEN1ALDH1A1
SCHEMBL21091915 0.76 DRD2 (0.59) CA1CA2ACHEMEN1ALDH1A1
SCHEMBL8019711 0.75 DRD2 (0.55)
SCHEMBL8978466 0.75 AGTR2 (0.44) CA1CA2ACHEMTNR1AMTNR1B
Hydrochloric Acid SCHEMBL7335560 0.74 DRD2 (0.54)
Hydrochloric Acid SCHEMBL7335562 0.74 DRD2 (0.54)
SCHEMBL8593552 0.74 ADRB3 (0.45) AGTR2
SCHEMBL21091908 0.70 KMT2A (0.51) MEN1ALDH1A1KMT2ASGMS2PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0608568-B1 Aminocycloalkanobenzodioxoles as beta-3 selective adrenergic agents AMERICAN CYANAMID CO (US) 1998-03-11 EP disclosed
US-5594027-A TREATMENT OF DIABETES, HYPERGLYCEMIA AND OBESITY AMERICAN CYANAMID COMPANY (US) 1997-01-14 US disclosed
US-5510376-A TREATING DIABETES, HYPERGLYCEMIA, OBESITY AMERICAN CYANAMID COMPANY (US) 1996-04-23 US disclosed
EP-0608568-A1 Aminocycloalkanobenzodioxoles as beta-3 selective adrenergic agents AMERICAN CYANAMID COMPANY (US) 1994-08-03 EP disclosed