SCHEMBL8548836

SCHEMBL8548836

CCN(CCO)CCOc1ccc2nc(CC(C)C)sc2c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.56
CYP1A2 P05177 1/20 0.55
CYP2D6 P10635 1/20 0.55
LSS P48449 2/20 0.45
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA4 P22748 1/20 0.42
HTT P42858 1/20 0.40
TSHR P16473 2/20 0.39
ALDH1A1 P00352 2/20 0.39
KMT2A Q03164 2/20 0.39
TP53 P04637 1/20 0.39
CYP3A4 P08684 1/20 0.39
HSD17B10 Q99714 1/20 0.39
PPARA Q07869 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ACHE P22303 1/20 0.39
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8550339 0.84 LMNA (0.55) LMNACYP1A2CYP2D6LSSCA1
SCHEMBL8361490 0.82 LMNA (0.53) LMNACYP1A2CYP2D6LSSCA1
SCHEMBL8552900 0.82 LMNA (0.53) LMNACYP1A2CYP2D6LSSCA1
SCHEMBL8361489 0.81 LMNA (0.52) LMNACYP1A2CYP2D6LSSCA1
SCHEMBL8552033 0.81 LMNA (0.52) LMNACYP1A2CYP2D6LSSCA1
SCHEMBL8357719 0.81 LMNA (0.58) LMNACYP1A2CYP2D6LSSCA1
SCHEMBL8551954 0.79 LMNA (0.50) LMNACYP1A2CYP2D6LSSCA1
SCHEMBL8551252 0.79 LMNA (0.50) LMNACYP1A2CYP2D6LSSCA1
SCHEMBL8356718 0.77 THRB (0.39) LMNATSHRALDH1A1KMT2ATP53
SCHEMBL8361945 0.76 LMNA (0.51) LMNACYP1A2CYP2D6LSSHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0824529-A1 BENZOTHIAZOLES AND BENZOXAZOLES, AS WELL AS DRUGS CONTAINING THEM, THEIR USE AND METHODS OF PREPARING THEM Dr. Karl Thomae GmbH (DE) 1998-02-25 EP disclosed
WO-1996035681-A1 BENZOTHIAZOLES AND BENZOXAZOLES, AS WELL AS DRUGS CONTAINING THEM, THEIR USE AND METHODS OF PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-11-14 WO disclosed