SCHEMBL8551954

SCHEMBL8551954

CCN(CCO)CCOc1ccc2nc(Cc3cccc4ccccc34)sc2c1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.50
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
LSS P48449 2/20 0.42
CDYL Q9Y232 1/20 0.41
ALK Q9UM73 2/20 0.39
KDM4E B2RXH2 1/20 0.39
HTR1D P28221 1/20 0.39
HTR1B P28222 1/20 0.39
PTPN1 P18031 1/20 0.38
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA4 P22748 1/20 0.37
ATP4A P20648 1/20 0.37
ATP4B P51164 1/20 0.37
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8357474 0.93 LMNA (0.57) LMNACYP1A2CYP2D6CDYLALK
SCHEMBL8552033 0.83 LMNA (0.52) LMNACYP1A2CYP2D6LSSALK
SCHEMBL8358150 0.82 RAB9A (0.41) LMNACYP1A2CYP2D6KDM4ECA1
SCHEMBL8358024 0.81 HTR1B (0.47) CDYLKDM4EHTR1DHTR1BPTPN1
SCHEMBL8361490 0.80 LMNA (0.53) LMNACYP1A2CYP2D6LSSCA1
SCHEMBL8552900 0.80 LMNA (0.53) LMNACYP1A2CYP2D6LSSCA1
SCHEMBL8548836 0.79 LMNA (0.56) LMNACYP1A2CYP2D6LSSKDM4E
SCHEMBL8550339 0.79 LMNA (0.55) LMNACYP1A2CYP2D6LSSCA1
SCHEMBL8358060 0.78 LMNA (0.63) LMNACYP1A2CYP2D6CA1CA2
SCHEMBL8551252 0.78 LMNA (0.50) LMNACYP1A2CYP2D6LSSCA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0824529-A1 BENZOTHIAZOLES AND BENZOXAZOLES, AS WELL AS DRUGS CONTAINING THEM, THEIR USE AND METHODS OF PREPARING THEM Dr. Karl Thomae GmbH (DE) 1998-02-25 EP disclosed
WO-1996035681-A1 BENZOTHIAZOLES AND BENZOXAZOLES, AS WELL AS DRUGS CONTAINING THEM, THEIR USE AND METHODS OF PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-11-14 WO disclosed