SCHEMBL8552033

SCHEMBL8552033

CCN(CCO)CCOc1ccc2nc(Cc3ccccn3)sc2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.52
CYP1A2 P05177 2/20 0.51
CYP2D6 P10635 2/20 0.51
LSS P48449 2/20 0.42
MAPT P10636 2/20 0.41
KMT2A Q03164 2/20 0.41
NPC1 O15118 1/20 0.41
PKM P14618 1/20 0.41
OPRK1 P41145 1/20 0.41
RAB9A P51151 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
ALK Q9UM73 1/20 0.39
CA4 P22748 1/20 0.39
ATP4A P20648 3/20 0.38
ATP4B P51164 3/20 0.38
HTT P42858 3/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8551954 0.83 LMNA (0.50) LMNACYP1A2CYP2D6LSSCA1
SCHEMBL8552900 0.82 LMNA (0.53) LMNACYP1A2CYP2D6LSSMAPT
SCHEMBL8361490 0.82 LMNA (0.53) LMNACYP1A2CYP2D6LSSMAPT
SCHEMBL8357948 0.81 NPC1 (0.42) LMNACYP1A2CYP2D6MAPTKMT2A
SCHEMBL8548836 0.81 LMNA (0.56) LMNACYP1A2CYP2D6LSSMAPT
SCHEMBL8550339 0.80 LMNA (0.55) LMNACYP1A2CYP2D6LSSKMT2A
SCHEMBL8355802 0.80 HTR1B (0.39) LMNAMAPTKMT2ANPC1PKM
SCHEMBL8358060 0.79 LMNA (0.63) LMNACYP1A2CYP2D6MAPTCA1
SCHEMBL8551252 0.79 LMNA (0.50) LMNACYP1A2CYP2D6LSSMAPT
SCHEMBL8357496 0.78 DRD2 (0.53) CYP1A2CYP2D6MAPTKMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0824529-A1 BENZOTHIAZOLES AND BENZOXAZOLES, AS WELL AS DRUGS CONTAINING THEM, THEIR USE AND METHODS OF PREPARING THEM Dr. Karl Thomae GmbH (DE) 1998-02-25 EP disclosed
WO-1996035681-A1 BENZOTHIAZOLES AND BENZOXAZOLES, AS WELL AS DRUGS CONTAINING THEM, THEIR USE AND METHODS OF PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-11-14 WO disclosed