SCHEMBL8549067

SCHEMBL8549067

N#Cc1cc(Oc2ccnc(Cl)c2)nc(-c2cccc(C(F)(F)F)c2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 6/20 0.45
CTSK P43235 11/20 0.43
KCNH2 Q12809 7/20 0.40
KDM4E B2RXH2 1/20 0.40
GRM5 P41594 1/20 0.39
KMO O15229 1/20 0.39
CTSB P07858 2/20 0.37
CTSL P07711 1/20 0.37
SCN9A Q15858 1/20 0.37
P2RY1 P47900 1/20 0.36
CCNA2 P20248 1/20 0.36
CDK2 P24941 1/20 0.36
CDK5 Q00535 1/20 0.36
DYRK1A Q13627 1/20 0.36
CDK5R1 Q15078 1/20 0.36
DYRK2 Q92630 1/20 0.36
DYRK1B Q9Y463 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8553275 0.89 GRM5 (0.41) CTSSCTSKKCNH2GRM5
SCHEMBL7009339 0.84 KMO (0.47) CTSSKDM4EKMOCCNA2CDK2
SCHEMBL8471818 0.81 PSD (0.41) CTSSKDM4EP2RY1CYP1A2CYP2C9
SCHEMBL8548872 0.79 POLB (0.43) CTSSCTSKKDM4ESCN9AP2RY1
SCHEMBL8552730 0.77 POLB (0.41) CTSSCTSKKDM4EP2RY1CYP1A2
SCHEMBL8553832 0.77 TRPV1 (0.43) CTSSCTSKKDM4ESCN9A
SCHEMBL8547908 0.76 POLB (0.41) CTSSCTSKKDM4ESCN9AP2RY1
SCHEMBL8773215 0.76 CYP1A2 (0.50) CTSSKDM4EP2RY1CYP1A2CYP2C9
SCHEMBL8546808 0.76 POLB (0.43) CTSSCTSKKDM4ESCN9AP2RY1
SCHEMBL8552758 0.75 KIF11 (0.42) CTSSCTSKKCNH2SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0820996-A1 Herbicidal cyanopyridines American Cyanamid Company (US) 1998-01-28 EP claimed
EP-0820996-A1 Herbicidal cyanopyridines American Cyanamid Company (US) 1998-01-28 EP disclosed