SCHEMBL8551012

SCHEMBL8551012

CCC(O)CC(c1cccnc1)c1ccc2cc(OC)ccc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 1/20 0.47
AKR1C3 P42330 3/20 0.47
AKR1C2 P52895 3/20 0.47
AKR1C1 Q04828 1/20 0.47
PTGS1 P23219 1/20 0.47
CYP11B2 P19099 8/20 0.46
CYP11B1 P15538 7/20 0.46
CYP17A1 P05093 4/20 0.46
CYP19A1 P11511 2/20 0.46
CYP2C9 P11712 1/20 0.46
KCNA5 P22460 1/20 0.43
CYP3A4 P08684 3/20 0.43
CYP2D6 P10635 2/20 0.43
SLC6A2 P23975 2/20 0.43
SLC6A4 P31645 2/20 0.43
SLC6A3 Q01959 2/20 0.43
KCNH2 Q12809 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
ABCB11 O95342 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8550178 0.89 PDE4D (0.42) PDE4DAKR1C3AKR1C2AKR1C1PTGS1
Hydrochloric Acid SCHEMBL8555644 0.85 CYP3A4 (0.44) PDE4DCYP11B2CYP11B1CYP17A1CYP19A1
SCHEMBL5752462 0.80 CYP11B2 (0.55) CYP11B2CYP11B1CYP17A1CYP19A1CYP2C9
SCHEMBL8551240 0.76 SMN1; SMN2 (0.44) PDE4DCYP17A1KCNA5SLC6A2SLC6A4
Ammonia Solution, Strong SCHEMBL6000232 0.75 KCNA5 (0.56) PDE4DCYP11B2CYP11B1CYP17A1CYP19A1
Ammonia Solution, Strong SCHEMBL5999968 0.74 CYP17A1 (0.61) PDE4DCYP17A1CYP19A1KCNA5SLC6A2
SCHEMBL7817339 0.74 CYP11B2 (0.50) CYP11B2CYP11B1CYP17A1CYP19A1CYP2C9
SCHEMBL8550753 0.72 TBXAS1 (0.45) PDE4DCYP2C9NPC1RAB9A
SCHEMBL8553222 0.71 PDE4D (0.49) PDE4DAKR1C3AKR1C2AKR1C1PTGS1
SCHEMBL8477516 0.70 CYP11B2 (0.51) CYP11B2CYP11B1CYP17A1CYP19A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865431-A2 COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-09-23 EP disclosed
WO-1997020815-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-06-12 WO disclosed