SCHEMBL8551360

SCHEMBL8551360

Cc1nc(Sc2ccc(C(=O)O)cn2)sc1CC(=O)O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
HPGD P15428 1/20 0.46
CYP2C19 P33261 1/20 0.46
HSD17B10 Q99714 1/20 0.46
RXRA P19793 1/20 0.41
RXRB P28702 1/20 0.41
RXRG P48443 1/20 0.41
KDM4E B2RXH2 2/20 0.40
CXCR2 P25025 1/20 0.38
TP53 P04637 2/20 0.36
MAPT P10636 1/20 0.36
HCAR3 P49019 5/20 0.36
HCAR2 Q8TDS4 1/20 0.36
P4HA1 P13674 2/20 0.36
P4HTM Q9NXG6 2/20 0.36
PPARG P37231 1/20 0.35
PPARD Q03181 1/20 0.35
PPARA Q07869 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8546628 0.89 ALDH1A1 (0.42) ALDH1A1CYP1A2CYP2C9HPGDCYP2C19
SCHEMBL8550265 0.82 PPARD (0.49) ALDH1A1KDM4EPPARGPPARDPPARA
SCHEMBL8591219 0.82 KDM5B (0.44) ALDH1A1KDM4EMAPTPPARGPPARD
SCHEMBL8545353 0.80 KDM4E (0.45) ALDH1A1CYP1A2HPGDHSD17B10KDM4E
SCHEMBL8673850 0.79 ALDH1A1 (0.41) ALDH1A1CYP1A2CYP2C9CYP2C19KDM4E
SCHEMBL8591973 0.77 ECE1 (0.42) ALDH1A1CYP1A2KDM4EPOLBPTGDR2
SCHEMBL8548708 0.76 PTGDR2 (0.40) ALDH1A1HPGDKDM4EMAPTPPARG
SCHEMBL10690460 0.75 LMNA (0.54) ALDH1A1HPGDKDM4EMAPTPOLB
SCHEMBL4481950 0.75 PTGDR2 (0.42) ALDH1A1CYP1A2KDM4EMAPTPPARD
SCHEMBL11588944 0.74 MAPT (0.43) ALDH1A1KDM4EMAPTGAAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0714393-B1 THIAZOLES AS ANTIVIRAL PFIZER (US) 1998-09-23 EP disclosed
US-5789408-A Antiviral thiazoles PFIZER INC. (US) 1998-08-04 US disclosed
EP-0714393-A1 THIAZOLES AS ANTIVIRAL PFIZER INC. (US) 1996-06-05 EP disclosed
WO-1995005378-A1 ANTIVIRAL THIAZOLES PFIZER INC. (US) 1995-02-23 WO disclosed