SCHEMBL8551467

SCHEMBL8551467

Cc1sc2ccc(NC(=O)c3cccc(I)c3)cc2c1CCN(C)Cc1cnco1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.36
IMPDH2 P12268 4/20 0.34
ROCK2 O75116 3/20 0.34
NAMPT P43490 1/20 0.33
KDR P35968 1/20 0.33
TP53 P04637 2/20 0.33
MAPT P10636 2/20 0.33
HTR1F P30939 1/20 0.32
BRAF P15056 1/20 0.32
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
PKM P14618 1/20 0.32
RAB9A P51151 1/20 0.32
NT5E P21589 1/20 0.32
PARP1 P09874 1/20 0.32
PTPN1 P18031 1/20 0.32
AURKA O14965 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8549783 0.85 GRM5 (0.37) GRM5IMPDH2ROCK2NAMPTKDR
SCHEMBL8191280 0.84 HTR1F (0.50) GRM5MAPTHTR1FALDH1A1LMNA
SCHEMBL5906312 0.75 HTR1F (0.51) GRM5HTR1FKDM4ENPC1ALDH1A1
SCHEMBL8551891 0.69 HTR1F (0.49) ROCK2NAMPTKDRTP53MAPT
Cadaverine Tartrate SCHEMBL8551708 0.68 MAP1LC3B (0.36) MAPTBRAFKDM4E
Benzoic Acid SCHEMBL8704380 0.66 TRPV1 (0.44) ROCK2TP53MAPTBRAFNPC1
Malonic Acid SCHEMBL8548925 0.66 HTR1F (0.47) NAMPTKDRTP53MAPTHTR1F
SCHEMBL8550328 0.65 FLT1 (0.37) KDRTP53MAPTHTR1FNPC1
Benzoic Acid SCHEMBL8548987 0.65 NPC1 (0.35) TP53MAPTNPC1ALDH1A1LMNA
SCHEMBL5785469 0.64 TRPV1 (0.64) GRM5TP53MAPTKDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0835869-A2 New serotonin 5-HT1F agonists ELI LILLY AND COMPANY (US) 1998-04-15 EP disclosed