SCHEMBL8551665

SCHEMBL8551665

CN(CCO)CCOc1ccc2nc(Cc3ccc(C(F)(F)F)cc3)sc2c1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 8/20 0.47
CACNA1H O95180 3/20 0.47
MAPT P10636 2/20 0.43
LMNA P02545 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
AURKA O14965 1/20 0.41
RPS6KB1 P23443 1/20 0.41
PPARG P37231 1/20 0.40
PPARD Q03181 1/20 0.40
PPARA Q07869 1/20 0.40
CSNK1D P48730 1/20 0.39
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA4 P22748 1/20 0.39
AURKB Q96GD4 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8551381 0.90 CACNA1B (0.45) CACNA1BCACNA1HMAPTLMNACYP1A2
SCHEMBL8357758 0.89 MAPT (0.44) CACNA1BMAPTLMNACYP1A2CYP2D6
SCHEMBL8359111 0.89 CACNA1B (0.53) CACNA1BCACNA1HMAPTLMNACYP1A2
SCHEMBL8551252 0.89 LMNA (0.50) CACNA1BCACNA1HMAPTLMNACYP1A2
SCHEMBL8355859 0.87 AURKB (0.49) MAPTLMNACYP1A2CYP2D6PPARD
SCHEMBL8550957 0.87 CACNA1B (0.44) CACNA1BCACNA1HMAPTLMNACYP1A2
SCHEMBL8361619 0.82 AURKB (0.46) MAPTLMNACYP1A2CYP2D6PPARD
SCHEMBL8516569 0.81 MAPT (0.44) CACNA1BCACNA1HMAPTLMNACYP1A2
SCHEMBL8358041 0.81 KMT2A (0.52) MAPTLMNACYP1A2CYP2D6PPARA
SCHEMBL8359679 0.79 MAPT (0.61) MAPTCYP1A2CSNK1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0824529-A1 BENZOTHIAZOLES AND BENZOXAZOLES, AS WELL AS DRUGS CONTAINING THEM, THEIR USE AND METHODS OF PREPARING THEM Dr. Karl Thomae GmbH (DE) 1998-02-25 EP disclosed
WO-1996035681-A1 BENZOTHIAZOLES AND BENZOXAZOLES, AS WELL AS DRUGS CONTAINING THEM, THEIR USE AND METHODS OF PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-11-14 WO disclosed