SCHEMBL8359111

SCHEMBL8359111

CN(C)CCOc1ccc2nc(Cc3ccc(C(F)(F)F)cc3)sc2c1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 7/20 0.53
CACNA1H O95180 3/20 0.53
LMNA P02545 1/20 0.46
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45
MAPT P10636 2/20 0.45
AURKB Q96GD4 1/20 0.44
LTA4H P09960 1/20 0.41
PPARG P37231 1/20 0.41
PPARD Q03181 1/20 0.41
PPARA Q07869 1/20 0.41
AURKA O14965 1/20 0.41
RPS6KB1 P23443 1/20 0.41
CSNK1D P48730 1/20 0.40
HRH3 Q9Y5N1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8551665 0.89 CACNA1B (0.47) CACNA1BCACNA1HLMNACYP1A2CYP2D6
SCHEMBL8357917 0.88 HTT (0.48) CACNA1BCACNA1HLMNACYP1A2CYP2D6
SCHEMBL8550957 0.87 CACNA1B (0.44) CACNA1BCACNA1HLMNACYP1A2CYP2D6
SCHEMBL8551381 0.87 CACNA1B (0.45) CACNA1BCACNA1HLMNACYP1A2CYP2D6
SCHEMBL8516569 0.86 MAPT (0.44) CACNA1BCACNA1HLMNACYP1A2CYP2D6
SCHEMBL8358041 0.85 KMT2A (0.52) LMNACYP1A2CYP2D6MAPTPPARA
SCHEMBL8355838 0.85 LTA4H (0.56) LMNACYP1A2CYP2D6MAPTAURKB
SCHEMBL8551252 0.85 LMNA (0.50) CACNA1BCACNA1HLMNACYP1A2CYP2D6
SCHEMBL8359679 0.83 MAPT (0.61) CYP1A2MAPTCSNK1D
SCHEMBL8554328 0.81 LMNA (0.48) CACNA1BCACNA1HLMNACYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5919807-A ANTICHOLESTEROL AGENTS DR. KARL THOMAE GMBH (DE) 1999-07-06 US disclosed
EP-0824529-A1 BENZOTHIAZOLES AND BENZOXAZOLES, AS WELL AS DRUGS CONTAINING THEM, THEIR USE AND METHODS OF PREPARING THEM Dr. Karl Thomae GmbH (DE) 1998-02-25 EP disclosed
WO-1996035681-A1 BENZOTHIAZOLES AND BENZOXAZOLES, AS WELL AS DRUGS CONTAINING THEM, THEIR USE AND METHODS OF PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-11-14 WO disclosed