SCHEMBL8551910

SCHEMBL8551910

O=C1NC(=O)C(c2ccccn2)(N2CCC(O)CC2)C(=O)N1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP3 P08254 1/20 0.46
MMP8 P22894 1/20 0.46
MMP2 P08253 12/20 0.42
MMP9 P14780 12/20 0.42
CHRM2 P08172 1/20 0.40
CHRM4 P08173 1/20 0.40
CHRM5 P08912 1/20 0.40
CHRM1 P11229 1/20 0.40
CHRM3 P20309 1/20 0.40
BRD4 O60885 1/20 0.39
GRIN1 Q05586 1/20 0.37
GRIN2A Q12879 1/20 0.37
GRIN2B Q13224 1/20 0.37
OPRM1 P35372 1/20 0.36
OPRL1 P41146 1/20 0.36
SLC6A9 P48067 1/20 0.36
ADAM17 P78536 1/20 0.36
ADAMTS5 Q9UNA0 1/20 0.36
CXCR3 P49682 1/20 0.35
HSD11B1 P28845 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8552412 0.80 MMP3 (0.40) MMP3MMP8MMP2MMP9BRD4
SCHEMBL27491360 0.79 MMP8 (0.69) MMP3MMP8MMP2MMP9BRD4
SCHEMBL8551083 0.79 MMP3 (0.44) MMP3MMP8MMP2MMP9BRD4
SCHEMBL8550568 0.77 MMP3 (0.52) MMP3MMP8MMP2MMP9BRD4
SCHEMBL8554743 0.75 MMP3 (0.51) MMP3MMP8MMP2MMP9CHRM2
SCHEMBL8551231 0.71 MMP3 (0.52) MMP3MMP8MMP2MMP9HSD11B1
SCHEMBL8550165 0.68 MMP8 (0.45) MMP3MMP8MMP2MMP9CHRM2
SCHEMBL8551269 0.66 MMP8 (0.49) MMP3MMP8MMP2MMP9BRD4
SCHEMBL8551832 0.65 MMP8 (0.65) MMP3MMP8MMP2MMP9
SCHEMBL743982 0.64 OPRM1 (0.51) CHRM2CHRM4CHRM5CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0869947-A1 NEW BARBITURIC ACID DERIVATIVES, PROCESSES FOR THEIR PRODUCTION AND PHARMACEUTICAL AGENTS CONTAINING THESE COMPOUNDS Roche Diagnostics GmbH (DE) 1998-10-14 EP disclosed
WO-1997023465-A1 NEW BARBITURIC ACID DERIVATIVES, PROCESSES FOR THEIR PRODUCTION AND PHARMACEUTICAL AGENTS CONTAINING THESE COMPOUNDS BOEHRINGER MANNHEIM GMBH (DE) 1997-07-03 WO disclosed