SCHEMBL8550319

SCHEMBL8550319

N=C(N)Nc1nnc(-c2ccccc2)c2cccc(C(F)(F)F)c12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.37
NPSR1 Q6W5P4 2/20 0.37
THRB P10828 1/20 0.37
PDE5A O76074 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
MAPT P10636 1/20 0.36
CYP2C9 P11712 1/20 0.36
HPGD P15428 1/20 0.36
ALOX15 P16050 1/20 0.36
CYP2C19 P33261 1/20 0.36
PDE1A P54750 1/20 0.36
PDE1B Q01064 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE1C Q14123 1/20 0.36
PDE3A Q14432 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8548628 0.99 KDM4E (0.37) KDM4ENPSR1THRBPDE5AALDH1A1
SCHEMBL8553708 0.91 LMNA (0.35) KDM4ENPSR1THRBMAPTSMN1; SMN2
SCHEMBL8547661 0.90 ALDH1A1 (0.43) NPSR1THRBALDH1A1MAPTHPGD
SCHEMBL8551148 0.85 ENPP3 (0.38) MAPTSMN1; SMN2CA9NR1H2NR1H3
SCHEMBL8374822 0.84 NPSR1 (0.39) KDM4ENPSR1THRBPDE5AALDH1A1
Hydrochloric Acid SCHEMBL8547376 0.82 NPSR1 (0.39) KDM4ENPSR1THRBPDE5AALDH1A1
SCHEMBL8552079 0.81 SMN1; SMN2 (0.34) KDM4ETHRBALDH1A1MAPTSMN1; SMN2
SCHEMBL8518196 0.81 NPSR1 (0.39) KDM4ENPSR1THRBPDE5AALDH1A1
Hydrochloric Acid SCHEMBL8549372 0.81 NPSR1 (0.39) KDM4ENPSR1THRBPDE5AALDH1A1
SCHEMBL8552267 0.80 HSD11B1 (0.38) KDM4ECYP1A2CYP3A4CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825187-A1 Condensed pyridazinyl guanidines, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-25 EP disclosed