SCHEMBL855227

SCHEMBL855227

COC(C)O[SiH2]c1ccccc1C

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.33
ACHE P22303 1/20 0.33
ESR1 P03372 1/20 0.32
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL706201 0.82 ACHE (0.38) TSHRACHEESR1SLC6A2SLC6A4
SCHEMBL22661034 0.79 CA2 (0.36) TSHR
SCHEMBL22661061 0.77 ADRA2A (0.36) TSHR
SCHEMBL3298602 0.75 CA4 (0.33)
SCHEMBL7935157 0.74 TSHR (0.43) TSHRACHEESR1
SCHEMBL28684438 0.74 ADRA2A (0.33)
SCHEMBL1314473 0.72 TSHR (0.32) TSHRACHEESR1
SCHEMBL713415 0.71 TRPA1 (0.35) TSHRSLC6A2SLC6A4SLC6A3
SCHEMBL11802576 0.70 TRPA1 (0.33)
SCHEMBL19927492 0.69 TSHR (0.33) TSHRACHEESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2476719-B1 IRREGULAR-SHAPED MICROPARTICLES, PROCESS FOR PRODUCTION OF IRREGULAR-SHAPED MICROPARTICLES, AND COSMETICS AND RESIN COMPOSITIONS CONTAINING IRREGULAR-SHAPED MICROPARTICLES TAKEMOTO OIL & FAT CO LTD (JP) 2019-01-02 EP disclosed
EP-2471841-B1 ORGANIC SILICONE PARTICLES, METHOD OF PRODUCING ORGANIC SILICONE PARTICLES, AND COSMETIC, RESIN COMPOSITION AND COATING COMPOSITION CONTAINING ORGANIC SILICONE PARTICLES TAKEMOTO OIL & FAT CO LTD (JP) 2014-07-30 EP disclosed
US-8524363-B2 Organosilicone fine particles of tetrahedral general shapes, method of production thereof and cosmetic materials, resin compositions and paint compositions containing same TAKEMOTO YUSHI KABUSHIKI KAISHA (JP) 2013-09-03 US disclosed
EP-2433979-B1 IRREGULAR-SHAPED HOLLOW MICROPARTICLE, METHOD FOR PRODUCING SAME, AND COSMETIC MATERIAL AND RESIN COMPOSITION CONTAINING IRREGULAR-SHAPED HOLLOW MICROPARTICLE TAKEMOTO OIL & FAT CO LTD (JP) 2013-06-12 EP disclosed
US-20130090411-A1 RESIN COMPOSITIONS CONTAINING NON-SPERICAL HOLLOW FINE PARTICLES ARATANI SATOSHI (JP) 2013-04-11 US disclosed
EP-2476719-A1 IRREGULAR-SHAPED MICROPARTICLES, PROCESS FOR PRODUCTION OF IRREGULAR-SHAPED MICROPARTICLES, AND COSMETICS AND RESIN COMPOSITIONS CONTAINING IRREGULAR-SHAPED MICROPARTICLES Takemoto Yushi Kabushiki Kaisha (JP) 2012-07-18 EP disclosed
EP-2471841-A1 ORGANIC SILICONE PARTICLES, METHOD OF PRODUCING ORGANIC SILICONE PARTICLES, AND COSMETIC, RESIN COMPOSITION AND COATING COMPOSITION CONTAINING ORGANIC SILICONE PARTICLES Takemoto Yushi Kabushiki Kaisha (JP) 2012-07-04 EP disclosed
EP-2433979-A1 IRREGULAR-SHAPED HOLLOW MICROPARTICLE, METHOD FOR PRODUCING SAME, AND COSMETIC MATERIAL AND RESIN COMPOSITION CONTAINING IRREGULAR-SHAPED HOLLOW MICROPARTICLE Takemoto Yushi Kabushiki Kaisha (JP) 2012-03-28 EP disclosed
US-20110224308-A1 ORGANOSILICONE FINE PARTICLES, METHOD OF PRODUCTION THEREOF AND COSMETIC MATERIALS, RESIN COMPOSITIONS AND PAINT COMPOSITIONS CONTAINING SAME TAKEMOTO YUSHI KABUSHIKI KAISHA (JP) 2011-09-15 US disclosed
US-20110171157-A1 NON-SPHERICAL FINE PARTICLES, METHOD OF PRODUCTION THEREOF AND COSMETIC MATERIALS AND RESIN COMPOSITIONS CONTAINING SAME ARATANI SATOSHI 2011-07-14 US disclosed
US-20110129672-A1 NON-SPHERICAL HOLLOW FINE PARTICLES, METHOD OF PRODUCTION THEREOF AND COSMETIC MATERIALS AND RESIN COMPOSITIONS CONTAINING SAME ARATANI SATOSHI 2011-06-02 US disclosed