SCHEMBL8552549

SCHEMBL8552549

Cc1cccc(C)c1NC(=O)CN1CCN(CC(=O)Nc2c(C)cccc2C)C(C(N)=O)C1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
KCNH2 Q12809 3/20 0.48
LMNA P02545 3/20 0.48
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
ADRB1 P08588 2/20 0.48
CYP3A4 P08684 2/20 0.48
ADRA2A P08913 2/20 0.48
CYP2D6 P10635 2/20 0.48
ADRA2B P18089 2/20 0.48
ADRA2C P18825 2/20 0.48
ADRA1A P35348 2/20 0.48
DRD3 P35462 2/20 0.48
HTR2B P41595 2/20 0.48
SLC29A1 Q99808 2/20 0.48
MLNR O43193 1/20 0.48
NR1I2 O75469 1/20 0.48
USP2 O75604 1/20 0.48
CYP1A2 P05177 1/20 0.48
PGR P06401 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10795286 0.87 KMT2A (0.57) ALDH1A1KCNH2LMNAMEN1KMT2A
SCHEMBL10680817 0.83 CYP3A4 (0.67) ALDH1A1KCNH2LMNAMEN1KMT2A
SCHEMBL10682648 0.82 LMNA (0.49) ALDH1A1KCNH2LMNAMEN1KMT2A
SCHEMBL10676648 0.82 ADRA1A (0.73) ALDH1A1KCNH2LMNAMEN1KMT2A
SCHEMBL10684438 0.80 CYP3A4 (0.58) ALDH1A1KCNH2LMNAMEN1KMT2A
SCHEMBL2327539 0.80 ALDH1A1 (0.64) ALDH1A1KCNH2LMNAMEN1KMT2A
SCHEMBL10680876 0.80 ALDH1A1 (0.43) ALDH1A1KCNH2LMNAMEN1KMT2A
SCHEMBL8554585 0.79 RXRA (0.43) LMNACYP3A4ADRA1ADRD3SLC29A1
SCHEMBL22407669 0.79 ALDH1A1 (0.52) ALDH1A1KCNH2LMNAMEN1KMT2A
Cadaverine Tartrate SCHEMBL10675929 0.78 ADRA1A (0.68) ALDH1A1KCNH2LMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0582164-B1 Adenosine re-uptake inhibiting derivatives of diphenyl oxazoles, thiazoles and imidazoles BRISTOL MYERS SQUIBB CO (US) 1998-12-23 EP disclosed
US-5382584-A Antiischemic agents BRISTOL-MYERS SQUIBB COMPANY (US) 1995-01-17 US disclosed
EP-0582164-A1 Adenosine re-uptake inhibiting derivatives of diphenyl oxazoles, thiazoles and imidazoles Bristol-Myers Squibb Company (US) 1994-02-09 EP disclosed