SCHEMBL8553033

SCHEMBL8553033

O=C(OC1CCN(Cc2ccccc2)CC1)c1ccc(Cl)cc1

nearest known ligand 0.70

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.70
DRD4 P21917 2/20 0.70
DRD3 P35462 1/20 0.60
BCHE P06276 3/20 0.60
LMNA P02545 1/20 0.59
POLB P06746 1/20 0.59
CHRM2 P08172 2/20 0.58
CHRM3 P20309 2/20 0.58
SIGMAR1 Q99720 1/20 0.55
CARM1 Q86X55 1/20 0.55
PRMT6 Q96LA8 1/20 0.55
ALDH1A1 P00352 1/20 0.53
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8551795 0.99 DRD2 (0.68) DRD2DRD4DRD3BCHELMNA
SCHEMBL8550706 0.95 DRD2 (0.62) DRD2DRD4DRD3BCHELMNA
Hydrochloric Acid SCHEMBL8552585 0.94 DRD2 (0.61) DRD2DRD4DRD3BCHELMNA
SCHEMBL8551065 0.93 DRD4 (0.60) DRD2DRD4DRD3BCHELMNA
Hydrochloric Acid SCHEMBL8550602 0.92 DRD2 (0.58) DRD2DRD4DRD3BCHELMNA
SCHEMBL8550490 0.92 BCHE (0.65) DRD2DRD4BCHECHRM2CHRM3
Hydrochloric Acid SCHEMBL8556315 0.91 MEN1 (0.65) DRD2DRD4BCHECHRM2CHRM3
SCHEMBL8552599 0.90 SIGMAR1 (0.64) DRD2DRD4BCHESIGMAR1
SCHEMBL8551087 0.88 SIGMAR1 (0.62) DRD2DRD4BCHESIGMAR1CARM1
SCHEMBL8550198 0.88 ADRB2 (0.57) DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1084329-C Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 2002-05-08 CN disclosed
EP-0871613-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 1998-10-21 EP disclosed
CN-1183768-A Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 1998-06-03 CN disclosed
US-5753679-A SCIZOPHRENIA HOFFMANN-LA ROCHE INC. (US) 1998-05-19 US disclosed
WO-1996035666-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 1996-11-14 WO disclosed