SCHEMBL8553724

SCHEMBL8553724

Nc1ccc(C(=O)OC2CCN(Cc3ccccc3)CC2)cc1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BCHE P06276 2/20 0.58
SIGMAR1 Q99720 2/20 0.57
OPRK1 P41145 1/20 0.56
DRD2 P14416 1/20 0.55
DRD4 P21917 1/20 0.55
CARM1 Q86X55 1/20 0.54
PRMT6 Q96LA8 1/20 0.54
SLC6A12 P48065 1/20 0.53
TMEM97 Q5BJF2 1/20 0.53
MCHR1 Q99705 1/20 0.53
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
SCN1A P35498 1/20 0.52
SCN2A Q99250 1/20 0.52
SCN3A Q9NY46 1/20 0.52
GAA P10253 1/20 0.52
KCNH2 Q12809 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8553941 0.95 CARM1 (0.57) BCHESIGMAR1OPRK1DRD2DRD4
Hydrochloric Acid SCHEMBL8555172 0.94 MEN1 (0.58) BCHESIGMAR1OPRK1DRD2DRD4
SCHEMBL8550490 0.91 BCHE (0.65) BCHEOPRK1DRD2DRD4CARM1
Hydrochloric Acid SCHEMBL8556315 0.89 MEN1 (0.65) BCHEOPRK1DRD2DRD4CARM1
SCHEMBL8553033 0.88 DRD2 (0.70) BCHESIGMAR1DRD2DRD4CARM1
SCHEMBL8552599 0.88 SIGMAR1 (0.64) BCHESIGMAR1DRD2DRD4SLC6A12
SCHEMBL8552222 0.88 SCN1A (0.60) SIGMAR1DRD4CARM1PRMT6MEN1
SCHEMBL8551087 0.87 SIGMAR1 (0.62) BCHESIGMAR1OPRK1DRD2DRD4
SCHEMBL8550662 0.87 SCN1A (0.63) BCHEDRD2DRD4CARM1PRMT6
SCHEMBL8549828 0.87 CHRM2 (0.59) BCHESIGMAR1DRD2DRD4CARM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1084329-C Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 2002-05-08 CN disclosed
EP-0871613-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 1998-10-21 EP disclosed
CN-1183768-A Benzyl piepridine derivs as pharmaceutical agents HOFFMANN LA ROCHE (CH) 1998-06-03 CN disclosed
US-5753679-A SCIZOPHRENIA HOFFMANN-LA ROCHE INC. (US) 1998-05-19 US disclosed
WO-1996035666-A1 BENZYL PIPERIDINE DERIVATIVES AS PHARMACEUTICAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 1996-11-14 WO disclosed