SCHEMBL8553771

SCHEMBL8553771

O=C1CC([S+]([O-])Cc2ccccc2)N1CCCOc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 3/20 0.44
SIGMAR1 Q99720 3/20 0.44
ALOX12 P18054 1/20 0.43
RAB9A P51151 5/20 0.41
SMN1; SMN2 Q16637 4/20 0.41
MAPT P10636 1/20 0.41
PLA2G7 Q13093 1/20 0.40
NPC1 O15118 3/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
HRH3 Q9Y5N1 2/20 0.39
POLB P06746 1/20 0.39
TSHR P16473 1/20 0.39
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 2/20 0.39
LMNA P02545 1/20 0.38
S1PR1 P21453 1/20 0.37
HTR1A P08908 1/20 0.36
DRD2 P14416 1/20 0.36
HTR2A P28223 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27499799 0.88 TEAD3 (0.40) MEN1KMT2AHRH3TSHRKDM4E
SCHEMBL8772495 0.85 GSK3A (0.41) SIGMAR1SMN1; SMN2MAPTMEN1KMT2A
SCHEMBL8772475 0.84 FAAH (0.42) SIGMAR1MEN1KMT2ATSHR
SCHEMBL8552234 0.84 PLA2G7 (0.46) TMEM97SIGMAR1ALOX12RAB9ASMN1; SMN2
SCHEMBL8439618 0.82 GSK3A (0.43) SIGMAR1MEN1KMT2ATSHR
SCHEMBL8772523 0.82 HCRTR1 (0.43) RAB9ASMN1; SMN2MAPTMEN1KMT2A
SCHEMBL8552101 0.81 LTA4H (0.39) MAPTMEN1KMT2ATSHRALDH1A1
SCHEMBL8550149 0.80 PKM (0.43) ALOX12RAB9ASMN1; SMN2NPC1MEN1
SCHEMBL8555803 0.80 HRH3 (0.41) SIGMAR1HRH3DRD2DRD3
SCHEMBL8440093 0.76 ITGB1 (0.39) SIGMAR1KMT2APOLBTSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0840725-A1 AZETIDINONE DERIVATIVES FOR THE TREATMENT OF ATHEROSCLEROSIS SMITHKLINE BEECHAM PLC (GB) 1998-05-13 EP claimed
WO-1997002242-A1 AZETIDINONE DERIVATIVES FOR THE TREATMENT OF ATHEROSCLEROSIS SMITHKLINE BEECHAM PLC (GB) 1997-01-23 WO claimed
EP-0840725-A1 AZETIDINONE DERIVATIVES FOR THE TREATMENT OF ATHEROSCLEROSIS SMITHKLINE BEECHAM PLC (GB) 1998-05-13 EP disclosed
WO-1997002242-A1 AZETIDINONE DERIVATIVES FOR THE TREATMENT OF ATHEROSCLEROSIS SMITHKLINE BEECHAM PLC (GB) 1997-01-23 WO disclosed