SCHEMBL8555698

SCHEMBL8555698

N#Cc1cnn(-c2ccccc2)c1NC(=O)NS(=O)(=O)c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 8/20 0.59
PTGS2 P35354 8/20 0.59
ALDH1A1 P00352 1/20 0.48
GFER P55789 1/20 0.47
MMP1 P03956 4/20 0.42
MMP2 P08253 4/20 0.42
MMP9 P14780 4/20 0.42
MMP8 P22894 4/20 0.42
MMP13 P45452 4/20 0.42
MAPT P10636 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
CA2 P00918 2/20 0.40
CA9 Q16790 2/20 0.40
CA1 P00915 1/20 0.40
CA4 P22748 1/20 0.40
POLB P06746 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
CA12 O43570 1/20 0.39
NPC1 O15118 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8559075 0.90 PTGS2 (0.63) PTGS1PTGS2ALDH1A1MMP1MMP2
SCHEMBL8551424 0.90 PTGS1 (0.65) PTGS1PTGS2GFERCA2CA9
SCHEMBL8552452 0.87 PTGS1 (0.62) PTGS1PTGS2ALDH1A1GFERMEN1
SCHEMBL8554553 0.87 PTGS2 (0.66) PTGS1PTGS2GFER
SCHEMBL8554524 0.87 PTGS1 (0.62) PTGS1PTGS2GFERMEN1KMT2A
SCHEMBL8553948 0.84 PTGS1 (0.62) PTGS1PTGS2GFERMAPT
SCHEMBL8556342 0.81 PTGS2 (0.72) PTGS1PTGS2ALDH1A1GFERKMT2A
SCHEMBL8551389 0.79 PTGS1 (0.51) PTGS1PTGS2ALDH1A1MEN1KMT2A
SCHEMBL8554179 0.79 PTGS1 (0.54) PTGS1PTGS2ALDH1A1GFERCA2
SCHEMBL8550834 0.77 PTGS2 (0.66) PTGS1PTGS2ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0885890-A1 SULFONYLUREIDOPYRAZOLE DERIVATIVES SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1998-12-23 EP disclosed