SCHEMBL8556935

SCHEMBL8556935

Cc1cccc(C)c1NC(=O)CN1CCN(Cc2nc(-c3ccccc3)c(-c3ccccc3)s2)CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
TSHR P16473 2/20 0.48
NPC1 O15118 1/20 0.48
CLK1 P49759 1/20 0.48
RAB9A P51151 1/20 0.48
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
KDR P35968 2/20 0.45
LMNA P02545 2/20 0.45
ADRB1 P08588 2/20 0.45
CYP3A4 P08684 2/20 0.45
ADRA2A P08913 2/20 0.45
CYP2D6 P10635 2/20 0.45
ADRA2B P18089 2/20 0.45
ADRA2C P18825 2/20 0.45
ADRA1A P35348 2/20 0.45
DRD3 P35462 2/20 0.45
HTR2B P41595 2/20 0.45
KCNH2 Q12809 2/20 0.45
MLNR O43193 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8552910 0.88 LMNA (0.50) ALDH1A1TSHRNPC1CLK1RAB9A
SCHEMBL8552887 0.80 NR4A2 (0.47) ALDH1A1TSHRMEN1KMT2AKDR
SCHEMBL6277857 0.79 MEN1 (0.65) ALDH1A1TSHRMEN1KMT2ALMNA
SCHEMBL8556067 0.78 CACNA1G (0.51) ALDH1A1TSHRMEN1KMT2AKDR
Hydrochloric Acid SCHEMBL8557858 0.77 CACNA1G (0.49) ALDH1A1TSHRMEN1KMT2AKDR
SCHEMBL2327539 0.76 ALDH1A1 (0.64) ALDH1A1TSHRMEN1KMT2ALMNA
SCHEMBL8556384 0.74 MEN1 (0.60) ALDH1A1TSHRMEN1KMT2ALMNA
SCHEMBL8555057 0.73 NR4A2 (0.51) TSHRMEN1KMT2ALMNAADRB1
SCHEMBL8557576 0.72 MEN1 (0.52) ALDH1A1TSHRMEN1KMT2ALMNA
SCHEMBL6261397 0.71 ALOX15 (0.74) ALDH1A1TSHRMEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0582164-B1 Adenosine re-uptake inhibiting derivatives of diphenyl oxazoles, thiazoles and imidazoles BRISTOL MYERS SQUIBB CO (US) 1998-12-23 EP claimed
US-5382584-A Antiischemic agents BRISTOL-MYERS SQUIBB COMPANY (US) 1995-01-17 US claimed
EP-0582164-A1 Adenosine re-uptake inhibiting derivatives of diphenyl oxazoles, thiazoles and imidazoles Bristol-Myers Squibb Company (US) 1994-02-09 EP claimed