SCHEMBL8558397

SCHEMBL8558397

Cn1cc2c(n1)-c1ccccc1N(C(=O)c1ccc([N+](=O)[O-])cc1)CC2

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.47
HPGD P15428 3/20 0.47
RAB9A P51151 3/20 0.47
AVPR2 P30518 1/20 0.46
AVPR1A P37288 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.45
KMT2A Q03164 2/20 0.45
ALDH1A1 P00352 2/20 0.45
NPC1 O15118 2/20 0.45
MAPT P10636 2/20 0.45
AR P10275 1/20 0.43
MEN1 O00255 1/20 0.43
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8559724 0.85 AVPR2 (0.51) SMN1; SMN2HPGDRAB9AAVPR2AVPR1A
SCHEMBL8562104 0.81 HPGD (0.58) SMN1; SMN2HPGDRAB9AL3MBTL1KMT2A
SCHEMBL5236488 0.81 AVPR2 (0.49) SMN1; SMN2HPGDRAB9AAVPR2AVPR1A
SCHEMBL8561524 0.80 HPGD (0.46) SMN1; SMN2HPGDRAB9AAVPR2AVPR1A
SCHEMBL6994753 0.80 AVPR2 (0.45) SMN1; SMN2HPGDRAB9AAVPR2AVPR1A
SCHEMBL7352575 0.78 ALDH1A1 (0.56) HPGDRAB9AL3MBTL1ALDH1A1NPC1
SCHEMBL21160915 0.78 HPGD (0.49) SMN1; SMN2HPGDRAB9AL3MBTL1KMT2A
SCHEMBL8561256 0.77 HPGD (0.48) SMN1; SMN2HPGDRAB9AL3MBTL1KMT2A
SCHEMBL8820731 0.77 AVPR1A (0.63) AVPR2AVPR1A
SCHEMBL8819120 0.77 AVPR2 (0.75) AVPR2AVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed
WO-1997047625-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS AMERICAN CYANAMID COMPANY (US) 1997-12-18 WO disclosed
WO-1997047624-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS AMERICAN CYANAMID COMPANY (US) 1997-12-18 WO disclosed
EP-0640592-A1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID COMPANY (US) 1995-03-01 EP disclosed