SCHEMBL8561256

SCHEMBL8561256

O=C(c1ccc([N+](=O)[O-])cc1)N1CCc2cnoc2-c2ccccc21

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.48
L3MBTL1 Q9Y468 1/20 0.47
P2RX4 Q99571 1/20 0.45
ALDH1A1 P00352 3/20 0.44
MAPT P10636 3/20 0.44
NPC1 O15118 2/20 0.44
LMNA P02545 1/20 0.44
HTT P42858 1/20 0.44
RAB9A P51151 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
STING1 Q86WV6 1/20 0.43
PDE4B Q07343 1/20 0.42
PDE4D Q08499 1/20 0.42
BCHE P06276 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8561104 0.84 AVPR2 (0.53) HPGDL3MBTL1P2RX4ALDH1A1NPC1
SCHEMBL8562104 0.83 HPGD (0.58) HPGDL3MBTL1ALDH1A1MAPTNPC1
SCHEMBL7352575 0.79 ALDH1A1 (0.56) HPGDL3MBTL1P2RX4ALDH1A1MAPT
SCHEMBL8561524 0.78 HPGD (0.46) HPGDL3MBTL1ALDH1A1MAPTNPC1
SCHEMBL8558397 0.77 SMN1; SMN2 (0.47) HPGDL3MBTL1ALDH1A1MAPTNPC1
SCHEMBL6990464 0.76 ALDH1A1 (0.52) HPGDL3MBTL1P2RX4ALDH1A1MAPT
SCHEMBL20599103 0.75 L3MBTL1 (0.48) HPGDL3MBTL1ALDH1A1MAPTNPC1
SCHEMBL7345718 0.75 ALDH1A1 (0.49) HPGDL3MBTL1P2RX4ALDH1A1MAPT
SCHEMBL19078673 0.75 L3MBTL1 (0.48) HPGDL3MBTL1ALDH1A1MAPTNPC1
SCHEMBL21160915 0.75 HPGD (0.49) HPGDL3MBTL1P2RX4ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed
WO-1997047625-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS AMERICAN CYANAMID COMPANY (US) 1997-12-18 WO disclosed
EP-0640592-A1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID COMPANY (US) 1995-03-01 EP disclosed