SCHEMBL8558815

SCHEMBL8558815

C[C@@H](N[C@@]1(CN)CCc2ccccc2C1)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 4/20 0.34
ALDH1A1 P00352 2/20 0.34
SIGMAR1 Q99720 2/20 0.33
CYP3A4 P08684 2/20 0.33
CHRM2 P08172 1/20 0.33
HTR1A P08908 1/20 0.33
ADRA2A P08913 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
CHRM1 P11229 1/20 0.33
SMPD1 P17405 1/20 0.33
DRD1 P21728 1/20 0.33
TBXA2R P21731 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
ADRA1A P35348 1/20 0.33
OPRM1 P35372 1/20 0.33
DRD3 P35462 1/20 0.33
CASR P41180 1/20 0.33
HTR2B P41595 1/20 0.33
SLC6A3 Q01959 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9180894 1.00 TAAR1 (0.34) TAAR1ALDH1A1SIGMAR1CYP3A4CHRM2
SCHEMBL12203625 0.77 HTR2A (0.37) TAAR1SIGMAR1ADRA2ASMN1; SMN2MEN1
SCHEMBL1587083 0.75 CYP3A4 (0.39) TAAR1ALDH1A1SIGMAR1CYP3A4CHRM2
SCHEMBL8557856 0.73 PLK1 (0.35) TAAR1ALDH1A1SIGMAR1GRM7SMN1; SMN2
SCHEMBL9260996 0.73 PLK1 (0.35) TAAR1ALDH1A1SIGMAR1GRM7SMN1; SMN2
SCHEMBL8556244 0.72 SIGMAR1 (0.41) ALDH1A1SIGMAR1CYP3A4CYP1A2CYP2D6
SCHEMBL9517420 0.71 HTR2A (0.37) TAAR1SIGMAR1ADRA2AOPRM1SMN1; SMN2
SCHEMBL31066736 0.67 MTOR (0.43) TAAR1CYP3A4GRM7ALOX15
SCHEMBL27899990 0.65 NPFFR1 (0.38) TAAR1CYP3A4LMNACYP1A2CYP2D6
SCHEMBL9519923 0.65 HTR2A (0.44) TAAR1SIGMAR1ADRA2ADRD1DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0635497-B1 Benzospiroalkene derivatives, process for their preparation and pharmaceutical compostions containing them ADIR (FR) 1998-05-20 EP disclosed
EP-0635497-A2 Benzospiroalkene derivatives, process for their preparation and pharmaceutical compostions containing them ADIR ET COMPAGNIE (FR) 1995-01-25 EP disclosed