SCHEMBL8559802

SCHEMBL8559802

COc1ccccc1-c1oc(Cc2ccccc2)nc1-c1ccccc1S(N)(=O)=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.49
SCN9A Q15858 1/20 0.41
GLA P06280 1/20 0.40
CA2 P00918 4/20 0.39
CA9 Q16790 4/20 0.39
CA12 O43570 3/20 0.38
CA1 P00915 3/20 0.38
PTGES2 Q9H7Z7 1/20 0.37
ALDH1A1 P00352 2/20 0.37
MAPT P10636 1/20 0.37
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
EGFR P00533 1/20 0.36
CCNT1 O60563 1/20 0.36
MAP4K4 O95819 1/20 0.36
CDK1 P06493 1/20 0.36
CDK4 P11802 1/20 0.36
CCNB1 P14635 1/20 0.36
CCNA2 P20248 1/20 0.36
CCND1 P24385 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8557954 0.96 RXRA (0.47) RXRASCN9AGLACA2CA9
SCHEMBL8556336 0.92 RXRA (0.41) RXRASCN9AGLACA2CA9
SCHEMBL8554229 0.91 CDK9 (0.42) RXRAGLACA2CA9CA12
SCHEMBL8553428 0.91 CA1 (0.42) RXRACA2CA9CA12CA1
SCHEMBL8559042 0.90 L3MBTL1 (0.43) RXRACA2CA9CA12CA1
SCHEMBL8555069 0.89 RXRA (0.43) RXRASCN9AGLACA2CA9
SCHEMBL8556147 0.89 MAPT (0.43) RXRASCN9ACA2CA9CA12
SCHEMBL8560691 0.88 CA1 (0.41) RXRACA2CA9CA12CA1
SCHEMBL8555338 0.87 RXRA (0.38) RXRASCN9AGLACA2CA9
SCHEMBL8560978 0.87 CDK9 (0.42) RXRACA2CA9CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719163-A ARTHRITIS G.D. SEARLE & CO. (US) 1998-02-17 US disclosed