SCHEMBL8553428

SCHEMBL8553428

COc1ccc(OC)c(-c2oc(Cc3ccccc3)nc2-c2ccccc2S(N)(=O)=O)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA9 Q16790 2/20 0.42
CA13 Q8N1Q1 1/20 0.42
RXRA P19793 1/20 0.41
ALDH1A1 P00352 5/20 0.40
P2RX3 P56373 4/20 0.40
EDNRA P25101 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
KDM4E B2RXH2 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
MAPK1 P28482 2/20 0.39
RECQL P46063 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
PTK2B Q14289 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8560691 0.97 CA1 (0.41) CA1CA2CA9CA13RXRA
SCHEMBL8559042 0.93 L3MBTL1 (0.43) CA1CA2CA9CA13RXRA
SCHEMBL8557664 0.91 L3MBTL1 (0.43) CA1CA2CA9CA13RXRA
SCHEMBL8559802 0.91 RXRA (0.49) CA1CA2CA9RXRAALDH1A1
SCHEMBL8557954 0.89 RXRA (0.47) CA1CA2CA9RXRAALDH1A1
SCHEMBL8556827 0.89 GRM2 (0.42) CA1CA2CA9CA13RXRA
SCHEMBL8555295 0.89 NR4A2 (0.36) CA1CA2CA9RXRAMAPT
SCHEMBL8556320 0.87 GRM2 (0.42) CA1CA2CA9RXRAALDH1A1
SCHEMBL8556976 0.87 SCN9A (0.44) RXRAALDH1A1L3MBTL1SMN1; SMN2MEN1
SCHEMBL8554223 0.87 GPR55 (0.36) CA1CA2CA9RXRAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719163-A ARTHRITIS G.D. SEARLE & CO. (US) 1998-02-17 US disclosed