SCHEMBL8560797

SCHEMBL8560797

O=C(Cl)c1ccc(F)c(C(=O)C(F)(F)F)c1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
ALOX15 P16050 1/20 0.41
PLA2G2D Q9UNK4 1/20 0.40
CES1 P23141 3/20 0.38
CES2 O00748 2/20 0.38
MLYCD O95822 3/20 0.34
ACHE P22303 2/20 0.34
MAPK1 P28482 1/20 0.33
KCNQ3 O43525 1/20 0.33
KCNQ2 O43526 1/20 0.33
KCNE1 P15382 1/20 0.33
KCNQ1 P51787 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8558758 0.84 PLA2G2D (0.55) PLA2G2DCES1CES2MAPK1
SCHEMBL11669995 0.83 ALDH1A1 (0.54) ALDH1A1ALOX15CES1CES2KCNQ3
SCHEMBL121698 0.79 TMPRSS4 (0.44) ALDH1A1CES1CES2
SCHEMBL15648925 0.79 LTA4H (0.44) ALDH1A1PLA2G2DCES1CES2MAPK1
SCHEMBL29470947 0.74 CES2 (0.67) ALDH1A1ALOX15CES1CES2KCNQ3
SCHEMBL192962 0.74 CES2 (0.67) ALDH1A1ALOX15CES1CES2KCNQ3
SCHEMBL7880210 0.74 CES1 (0.60) ALDH1A1CES1MLYCDACHE
SCHEMBL24166639 0.74 MAPT (0.41) ALDH1A1ALOX15PLA2G2DCES1CES2
SCHEMBL2966997 0.74 DGAT1 (0.47) ALDH1A1ALOX15CES1CES2
SCHEMBL759728 0.74 KCNQ3 (0.54) CES1CES2KCNQ3KCNQ2KCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5747541-A Substituted benzoylguanidines, a process for their preparation, their use as medicament of diagnostic agent, and medicament comprising them HOECHST AKTIENGESELLSCHAFT (DE) 1998-05-05 US disclosed