SCHEMBL8562079

SCHEMBL8562079

COc1cc(C(=O)N2c3ccccc3CNc3ccccc32)ccc1NC(=O)c1cc(F)ccc1C

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 14/20 0.47
AVPR1A P37288 13/20 0.47
TUBB4A P04350 1/20 0.41
TUBB P07437 1/20 0.41
TUBA3C P0DPH7 1/20 0.41
TUBA1B P68363 1/20 0.41
TUBA4A P68366 1/20 0.41
TUBB4B P68371 1/20 0.41
TUBB3 Q13509 1/20 0.41
TUBB2A Q13885 1/20 0.41
TUBB8 Q3ZCM7 1/20 0.41
TUBA3E Q6PEY2 1/20 0.41
TUBA1A Q71U36 1/20 0.41
TUBA1C Q9BQE3 1/20 0.41
TUBB6 Q9BUF5 1/20 0.41
TUBB2B Q9BVA1 1/20 0.41
TUBB1 Q9H4B7 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HSD11B1 P28845 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8560113 0.91 ALDH1A1 (0.51) AVPR2AVPR1ATUBB4ATUBBTUBA3C
SCHEMBL8557684 0.89 AVPR2 (0.51) AVPR2AVPR1ATUBB4ATUBBTUBA3C
SCHEMBL8563485 0.87 PYGL (0.42) AVPR2AVPR1ATUBB4ATUBBTUBA3C
SCHEMBL8558577 0.85 AVPR2 (0.57) AVPR2AVPR1A
SCHEMBL8556903 0.83 AVPR2 (0.53) AVPR2AVPR1ATUBB4ATUBBTUBA3C
SCHEMBL8562249 0.81 AVPR2 (0.45) AVPR2AVPR1ATUBB4ATUBBTUBA3C
SCHEMBL8556991 0.81 AVPR2 (0.58) AVPR2AVPR1A
SCHEMBL8561948 0.79 AVPR2 (0.51) AVPR2AVPR1A
SCHEMBL8557275 0.79 AVPR2 (0.59) AVPR2AVPR1A
SCHEMBL8558373 0.77 AVPR2 (0.59) AVPR2AVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed